drugset / Trial / NCT02705963

A Drug-Drug Interaction Study to Assess the Effect of Trametinib on the Pharmacokinetics of an Oral Contraceptive in Female Patients With Solid Tumors

NCT02705963

Phase 1 Completed 19 enrolled Novartis Pharmaceuticals
NaSingle-groupOpen-labelTreatment

Summary

The purpose of this study is to evaluate the effect of trametinib once daily on the pharmacokinetics (PK) of a daily dosing oral contraceptives (OCs) containing norethindrone (NE) and ethinyl estradiol (EE) in female patients with solid tumors. The PK of trametinib and its metabolite M5 will also be assessed.

Timeline

Start
2016-10-20
Primary completion
2019-08-29
Completion
2019-08-29

Drugs

EvaluationDrugModalityDoseRoute
Subject Norethindrone Unknown 1 mg Oral
Subject Trametinib Small molecule 0.5 mg Oral
Subject Trametinib Small molecule 2 mg Oral
Subject ethinyl estradiol Small molecule 0.035 mg Oral

Indications