drugset / Trial / NCT04142762

A Study to Assess CYP3A4 Modulator, Oral Contraceptive, and pH Modifier Drug Interactions for ABI-H2158 in Healthy Adults

NCT04142762

Phase 1 Completed 80 enrolled Assembly Biosciences
Non-randomizedParallel-groupOpen-labelTreatment

Summary

This study is designed to assess 1) the effect of multiple doses of itraconazole (CYP3A4 inhibitor), rifampin (CYP3A4 inducer), and esomeprazole (pH modifier) on the pharmacokinetics of a single oral dose of ABI-H2158, and 2) the effect of steady-state oral ABI-H2158 on the pharmacokinetics of midazolam (sedative) and levonorgestrel/ethinyl estradiol (active oral contraceptive) in healthy adult participants.

Timeline

Start
2019-10-18
Primary completion
2020-01-12
Completion
2020-01-29

Drugs

EvaluationDrugModalityDoseRoute
Subject ABI-H2158 Unknown Oral
Subject Esomeprazole Small molecule Oral
Subject Itraconazole Small molecule Oral
Subject Levonorgestrel Small molecule Oral
Subject Midazolam Small molecule Oral
Subject Rifampin Small molecule Oral
Subject ethinyl estradiol Small molecule Oral