drugset / Trial / NCT04166669

A Drug-Drug Interaction Study of CYP3A4 Inhibition and Pan-CYP Induction on APX001

NCT04166669

Phase 1 Completed 36 enrolled Basilea Pharmaceutica
Non-randomizedParallel-groupOpen-labelTreatment

Summary

This is a Phase 1, open-label study to evaluate the drug-drug interaction potential of a strong CYP3A4 inhibitor (itraconazole) and a pan-CYP inducer (rifampin) on APX001 in two parallel groups of healthy subjects.

Timeline

Start
2019-11-12
Primary completion
2020-03-03
Completion
2020-03-03

Drugs

EvaluationDrugModalityDoseRoute
Subject Fosmanogepix Small molecule 500 mg Intravenous
Subject Fosmanogepix Small molecule 1000 mg Intravenous
Subject Itraconazole Small molecule 200 mg Oral
Subject Rifampin Small molecule 600 mg Oral