drugset / Trial / NCT04997902

Combination Trial of Tipifarnib and Alpelisib in Adult Recurrent/ Metastatic Head and Neck Squamous Cell Carcinoma (R/M HNSCC)

NCT04997902

Phase 1/2 Completed 45 enrolled Kura Oncology, Inc.
Non-randomizedParallel-groupOpen-labelTreatment

Summary

This phase 1/2 combination trial of tipifarnib, a farnesyltransferase inhibitor, and alpelisib, a PI3K inhibitor in participants with recurrent/metastatic head and neck squamous cell carcinoma (HNSCC) whose tumors overexpress the HRAS protein and/or are PIK3CA-mutated and/or PIK3CA-amplified.

Timeline

Start
2021-12-07
Primary completion
2025-08-29
Completion
2025-08-29

Drugs

EvaluationDrugModalityDoseRoute
Subject Alpelisib Small molecule Oral
Subject tipifarnib Small molecule Oral