drugset / Trial / NCT05633979

Phase 1b Study of EZH1/2 Inhibitor Valemetostat in Combination With Trastuzumab Deruxtecan in Subjects With HER2 Low/Ultra-low/Null Metastatic Breast Cancer

NCT05633979

Phase 1 Active not recruiting 17 enrolled M.D. Anderson Cancer Center Daiichi Sankyo · collab
Non-randomizedSingle-groupOpen-labelTreatment

Summary

To find a recommended dose of valemetostat that can be given in combination with trastuzumab deruxtecan to patients with low/ultra-low HER2-expressing metastatic breast cancer.

Timeline

Start
2023-02-09
Primary completion
2030-12-31
Completion
2032-12-31

Drugs

EvaluationDrugModalityDoseRoute
Subject Trastuzumab deruxtecan Monoclonal antibody Intravenous
Subject Valemetostat Small molecule Oral

Indications