drugset / Trial / NCT06689527

Evaluation of Vamorolone CYP3A4 Induction on Midazolam (a Sensitive CYP 3A4 Substrate) Pharmacokinetics

NCT06689527

Phase 1 Completed 18 enrolled Santhera Pharmaceuticals
NaSingle-groupOpen-labelOther

Summary

The purpose of this study was to investigate how vamorolone affects the CYP3A4 enzyme in humans by measuring the pharmacokinetics of midazolam and its metabolite, 1'-hydroxymidazolam, in healthy subjects. The pharmacokinetics of midazolam were measured on Day 1 and then on Day 14 to investigate the potential interaction between the two compounds. The safety and the tolerability was also investigated.

Timeline

Start
2024-08-13
Primary completion
2024-09-24
Completion
2024-10-16

Drugs

EvaluationDrugModalityDoseRoute
Subject Midazolam Small molecule 2.5 mg Oral
Subject Vamorolone Small molecule 6 mg/kg Oral

Indications

No indication recorded.