Drugs / Treprostinil
last change Jun 2026 re-read 2 minutes ago

Treprostinil

Other / unclassified

Developed for
pulmonary arterial hypertension · pulmonary hypertension · chronic obstructive pulmonary disease · systemic sclerosis · idiopathic pulmonary fibrosis · interstitial lung disease · limb ischemia · pulmonary fibrosis
+17 more · pulmonary hypertension owing to lung disease and/or hypoxia · congenital heart disease · ischemic disease · peripheral vascular disease · pulmonary hypertension, primary, 6 · ulcer of lower limbs · calcinosis · chronic thromboembolic pulmonary hypertension · combined pulmonary fibrosis-emphysema syndrome · diastolic heart failure · polycythemia due to hypoxia · Raynaud disease · restless legs syndrome · sarcoidosis · univentricular heart · adult acute respiratory distress syndrome · pulmonary hypertension, neonatal
Investigated by
United Therapeutics · Liquidia Technologies, Inc. · University Hospital, Grenoble · Lung Biotechnology PBC · AOP Orphan Pharmaceuticals AG · CVie Therapeutics Co. Ltd.
+40 more · Eli Lilly and Company · Nuventra, Inc. · PPD Development, LP · Stanford University · ANOVA CRO s.r.o. · Abhinav Humar, MD · Aixial s.r.o. · Asian Clinical Trials · Bastiaan Driehuys · Bial - Portela C S.A. · Brigham and Women's Hospital · Children's Hospital Medical Center, Cincinnati · FGK Clinical Research GmbH · GCP-Service International Ltd. & Co. KG · Guangzhou Institute of Respiratory Disease · Jewish General Hospital · Linksium · Lundquist Institute for Biomedical Innovation at Harbor-UCLA Medical Center · Magdi H. Yacoub · Mannkind Corporation · Mayo Clinic · Ochsner Health System · PharmaLex Belgium · Pharmosa Biopharm Inc. · Rajan Saggar · Rhode Island Hospital · SciPharm SàRL · Shanghai Jiao Tong University School of Medicine · Shanghai Zhongshan Hospital · Southern Arizona Vascular Institute · Southern Illinois University · University Grenoble Alps · University of Alberta · University of Arizona · University of California, Los Angeles · University of California, San Diego · University of Colorado, Denver · University of Florida · University of Pittsburgh Medical Center · University of Rhode Island

Regulatory milestones approvals, filings & regulatory actions · 7 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (3) US (FDA) TYVASO 2014-05-20 – 2021-03-31 fda.gov
Approved EU (EMA) Trepulmix 2020-04-03 europa.eu
Label expansions (2) US (FDA) REMODULIN 2004-11-24 – 2006-03-20 fda.gov
Approved US (FDA) REMODULIN 2002-05-21 fda.gov

Trials 88 · started per year

today
US approved 2002
EU approved 2020
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1998199920002001200220032004200520062007200820092010201120122013201420152016201720182019202020212022202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT07116681 Oct 2025 → Jul 2027 expected pulmonary hypertension University of California, San Diego Not yet recruiting No outcome recorded
Phase 112 trials
Phase 1 NCT05067270 Oct → Dec 2021 type 1 diabetes mellitus Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT03950739 Sep 2019 → Aug 2023 pulmonary arterial hypertension United Therapeutics Completed No outcome recorded
Phase 1 NCT04041648 Nov 2018 → Sep 2019 pulmonary arterial hypertension Pharmosa Biopharm Inc. Completed No outcome recorded
Phase 1 NCT03464864 Mar → Jun 2018 pulmonary arterial hypertension Mannkind Corporation Completed No outcome recorded
Phase 1 NCT04675944 Feb → May 2018 pulmonary arterial hypertension Bial - Portela C S.A. Completed No outcome recorded
Phase 1 NCT02770521 May → Jul 2016 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01481974 Dec 2012 → May 2019 ischemic disease Abhinav Humar, MD Completed No outcome recorded
Phase 1 NCT01758744 Dec 2012 → Jul 2016 chronic obstructive pulmonary disease, pulmonary hypertension University of Colorado, Denver Completed No outcome recorded
Phase 1 NCT01746485 Jul 2012 United Therapeutics Completed No outcome recorded
Phase 1 NCT01172496 Aug 2010 pulmonary arterial hypertension United Therapeutics Completed No outcome recorded
Phase 1/25 trials
Phase 1/2 NCT04005469 Nov 2020 → Jun 2028 expected ischemic disease Rhode Island Hospital Recruiting No outcome recorded
Phase 1/2 NCT03654989 Jan 2020 → Dec 2021 ulcer of lower limbs University Hospital, Grenoble Terminated No outcome recorded
Phase 1/2 NCT03120533 Jun 2017 → Jun 2019 systemic sclerosis University Hospital, Grenoble Completed No outcome recorded
Phase 1/2 NCT01554540 Feb 2012 → Oct 2013 systemic sclerosis University Hospital, Grenoble Unknown No outcome recorded
Phase 1/2 NCT01082484 Jan 2010 → Jan 2011 University Hospital, Grenoble Completed No outcome recorded
Phase 220 trials
Phase 2 NCT07177703 Oct 2025 → Dec 2027 expected pulmonary arterial hypertension Shanghai Zhongshan Hospital Not yet recruiting No outcome recorded
Phase 2 NCT07037836 Sep 2025 → Jul 2027 expected chronic obstructive pulmonary disease, polycythemia due to hypoxia Bastiaan Driehuys Recruiting No outcome recorded
Phase 2 NCT06969573 Jun 2025 → Dec 2026 expected chronic obstructive pulmonary disease University of Alberta Active not recruiting No outcome recorded
Phase 2 NCT05564637 Mar 2023 → Oct 2024 interstitial lung disease, pulmonary arterial hypertension Mayo Clinic Completed No outcome recorded
Phase 2 NCT03814317 Jan 2020 → Dec 2025 interstitial lung disease, pulmonary hypertension, sarcoidosis University of Florida Completed No outcome recorded
Phase 2 NCT03884465 Nov 2019 → Dec 2020 pulmonary arterial hypertension Liquidia Technologies, Inc. Terminated No outcome recorded
Phase 2 NCT03016468 May 2017 → Sep 2018 pulmonary arterial hypertension United Therapeutics Withdrawn No outcome recorded
Phase 2 NCT03012646 Apr 2017 → Apr 2019 chronic obstructive pulmonary disease, pulmonary hypertension United Therapeutics Withdrawn No outcome recorded
Phase 2 NCT02769624 Feb 2017 → Sep 2018 congenital heart disease Children's Hospital Medical Center, Cincinnati Terminated No outcome recorded
Phase 2 NCT02663895 Oct 2016 → May 2020 calcinosis, systemic sclerosis Stanford University Completed No outcome recorded
Phase 2/33 trials
Phase 2/3 NCT02633293 Sep 2016 → Aug 2021 combined pulmonary fibrosis-emphysema syndrome, interstitial lung disease, pulmonary hypertension United Therapeutics Terminated No outcome recorded
Phase 2/3 NCT01884038 Jun 2008 → Jun 2010 United Therapeutics Withdrawn No outcome recorded
Phase 2/3 NCT00067041 Mar → Dec 2003 peripheral vascular disease United Therapeutics Terminated No outcome recorded
Phase 326 trials
Phase 3 NCT07285655 Apr 2026 → Jul 2029 expected pulmonary hypertension owing to lung disease and/or hypoxia Liquidia Technologies, Inc. Recruiting No outcome recorded
Phase 3 NCT06350032 Jul 2024 → Nov 2028 expected pulmonary arterial hypertension AOP Orphan Pharmaceuticals AG Recruiting No outcome recorded
Phase 3 NCT05943535 Oct 2023 → Nov 2027 expected pulmonary fibrosis United Therapeutics Recruiting No outcome recorded
Phase 3 NCT05255991 Oct 2022 → Jun 2025 idiopathic pulmonary fibrosis United Therapeutics Completed No outcome recorded
Phase 3 NCT04905693 Sep 2022 → Jun 2026 overdue idiopathic pulmonary fibrosis, pulmonary fibrosis United Therapeutics Enrolling by invitation No outcome recorded
Phase 3 NCT04691154 Aug 2021 → Mar 2025 overdue pulmonary arterial hypertension, pulmonary hypertension owing to lung disease and/or hypoxia Liquidia Technologies, Inc. Active not recruiting No outcome recorded
Phase 3 NCT04708782 Jun 2021 → Feb 2026 idiopathic pulmonary fibrosis United Therapeutics Completed No outcome recorded
Phase 3 NCT03992755 Jul 2019 → May 2025 overdue pulmonary hypertension, primary, 6 Liquidia Technologies, Inc. Active not recruiting No outcome recorded
Phase 3 NCT04062565 Mar 2019 → Dec 2025 overdue pulmonary arterial hypertension University of Arizona Recruiting No outcome recorded
Phase 3 NCT03794583 Dec 2018 → Nov 2022 chronic obstructive pulmonary disease, pulmonary hypertension United Therapeutics Terminated No outcome recorded
Phase 419 trials
Phase 4 NCT07112183 Oct 2025 → Sep 2028 expected Raynaud disease Brigham and Women's Hospital Recruiting No outcome recorded
Phase 4 NCT06317805 Dec 2023 → Jun 2027 expected pulmonary arterial hypertension AOP Orphan Pharmaceuticals AG Recruiting No outcome recorded
Phase 4 NCT05203510 Oct 2022 → Apr 2026 overdue pulmonary arterial hypertension United Therapeutics Active not recruiting No outcome recorded
Phase 4 NCT03835676 May 2019 → Jun 2025 pulmonary hypertension Magdi H. Yacoub Unknown No outcome recorded
Phase 4 NCT03497689 Jan 2019 → May 2022 pulmonary arterial hypertension United Therapeutics Completed No outcome recorded
Phase 4 NCT02882126 Jun 2017 → Jun 2021 pulmonary arterial hypertension United Therapeutics Withdrawn No outcome recorded
Phase 4 NCT02893995 Feb 2017 → Apr 2018 pulmonary arterial hypertension United Therapeutics Withdrawn No outcome recorded
Phase 4 NCT06605326 Jan 2015 → Sep 2024 heart failure, pulmonary arterial hypertension, pulmonary hypertension owing to lung disease and/or hypoxia Guangzhou Institute of Respiratory Disease Completed No outcome recorded
Phase 4 NCT01615627 Jul 2012 → Feb 2019 pulmonary arterial hypertension Jewish General Hospital Withdrawn No outcome recorded
Phase 4 NCT02847260 Apr 2012 → Mar 2014 pulmonary arterial hypertension United Therapeutics Completed No outcome recorded
Phase not applicable2 trials
NCT02498444 Sep 2015 → Dec 2020 univentricular heart Stanford University Terminated No outcome recorded
NCT01980979 Nov 2013 → Dec 2015 congenital heart disease University of California, Los Angeles Withdrawn No outcome recorded
Also used as a comparator or background therapy in 12 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT02583789 Comparator May 2016 → Dec 2021 Raynaud disease Brigham and Women's Hospital Completed No outcome recorded
Phase 11 trial
Phase 1 NCT06193031 Background Nov → Dec 2015 Insmed Incorporated Completed No outcome recorded
Phase 23 trials
Phase 2 NCT02178566 Comparator Aug 2015 → Jan 2019 chronic obstructive pulmonary disease Inova Health Care Services Terminated No outcome recorded
Phase 2 NCT02261883 Comparator Jul 2015 → Sep 2022 pulmonary hypertension, neonatal United Therapeutics Terminated No outcome recorded
Phase 2 NCT02370095 Comparator Feb 2015 → Oct 2017 adult acute respiratory distress syndrome University of North Carolina, Chapel Hill Terminated No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT02630316 Comparator Feb 2017 → Dec 2019 combined pulmonary fibrosis-emphysema syndrome, interstitial lung disease, pulmonary hypertension United Therapeutics Completed No outcome recorded
Phase 34 trials
Phase 3 NCT02999906 Comparator Oct 2017 → Dec 2021 pulmonary arterial hypertension United Therapeutics Withdrawn No outcome recorded
Phase 3 NCT00760916 Comparator Dec 2008 → Jan 2009 pulmonary hypertension United Therapeutics Withdrawn No outcome recorded
Phase 3 NCT00325403 Comparator Oct 2006 → Apr 2011 pulmonary hypertension United Therapeutics Completed No outcome recorded
Phase 3 NCT00325442 Comparator Oct 2006 → Sep 2008 pulmonary arterial hypertension United Therapeutics Completed No outcome recorded
Phase 41 trial
Phase 4 NCT01305252 Comparator Jul 2010 → Sep 2014 pulmonary arterial hypertension Stanford University Completed No outcome recorded
Phase not stated1 trial
NCT05572996 Background combined pulmonary fibrosis-emphysema syndrome, interstitial lung disease, pulmonary hypertension Ferrer Internacional S.A. Available No outcome recorded

Evidence & citations 17 cited values

Every value below carries the sentence it was read from. 103 sources stand behind the page.

FieldValueCited text
Known as treprostinil “This multi-center, open-label study will assess the tolerability and safety of transitioning subjects with stable Pulmonary Arterial Hypertension (PAH) from continuous...” NCT01588405
87

“The purpose of this multi-center, open-label, safety and tolerability study was to assess the addition of oral treprostinil (UT-15C sustained release \[SR\] tablets) to...” NCT01477333

“FREEDOM DR: Oral Treprostinil in Combination With an Endothelin Receptor Antagonist (ERA) and/or a Phosphodiesterase-5 (PDE-5) Inhibitor or as Monotherapy for the Treatment of...” NCT00760916

“Remodulin (treprostinil sodium), a prostacyclin analog, possesses potent pulmonary and systemic vasodilatory and platelet anti-aggregatory actions in vitro and in vivo.” NCT00458042

Treprostinil diolamine (oral treprostinil) is an orally available prostacyclin analog that was developed for the treatment of pulmonary arterial hypertension.” PMID 24603117 Mar 2014

Treprostinil is a stable prostacyclin analog approved for the treatment of pulmonary arterial hypertension (PAH) as parenteral or inhaled therapy.” PMID 23669822 Sep 2013

“Liposomal Treprostinil Inhalation Suspension (L606)” NCT04691154

NCT02882126

NCT03654989

NCT07112183

NCT04062565

NCT01560637

NCT02603068

NCT00848107

NCT01268553

NCT00848939

NCT02583789

NCT03496623

NCT05572996

NCT04005469

NCT01560624

NCT03794583

NCT05943535

NCT02999906

NCT00439946

NCT00445159

NCT00325403

NCT01305252

NCT00067041

NCT02498444

NCT01554540

NCT00060996

NCT03814317

NCT03497689

NCT05203510

NCT03835676

NCT06969573

NCT07037836

NCT03399604

NCT00651885

NCT00058929

NCT01172496

NCT06317805

NCT00741819

NCT01758744

NCT02769624

NCT00325442

NCT05067270

NCT06605326

NCT04041648

NCT04675944

NCT03884465

NCT07177703

NCT02633293

NCT03055221

NCT00494533

NCT02630316

NCT04708782

NCT02178566

NCT02770521

NCT00705133

NCT01027949

NCT05255991

NCT02893995

NCT01416636

NCT01131845

NCT03992755

NCT03043651

NCT00703339

NCT01481974

NCT02663895

NCT01082484

NCT01557647

NCT02276872

NCT01557660

NCT04905693

NCT03055234

NCT03016468

NCT03012646

NCT06350032

NCT03950739

NCT03120533

NCT00775463

NCT03464864

NCT01615627

NCT05564637

NCT02370095

NCT03037580

Known as Inhaled treprostinil ClinicalTrials.gov intervention name — accepted as the source's own label NCT00147199
1

NCT07116681

Known as iTRE “evaluated the safety and efficacy of inhaled treprostinil (iTRE) in this patient population.” PMID 38811045 Jun 2024
Known as L606 “The primary objective of this study is to evaluate the Pharmacokinetics, Safety and Tolerability of L606 (Liposomal Treprostinil) Inhalation Solution in Single Ascending Dose...” NCT04041648
2

“Liposomal Treprostinil Inhalation Suspension (L606)” NCT04691154

NCT07285655

Known as LIQ861 “Inhaled LIQ861 (Treprostinil) in Pulmonary Arterial Hypertension (WHO Group 1) Patients” NCT03992755
1

“inhaled dry powder treprostinil (LIQ861)” NCT03884465

Known as Remodulin Remodulin (treprostinil sodium), a prostacyclin analog, possesses potent pulmonary and systemic vasodilatory and platelet anti-aggregatory actions in vitro and in vivo.” NCT00458042
8

Remodulin® (treprostinil sodium), a stable analogue of prostacyclin” NCT00643604

Remodulin® (treprostinil sodium) Injection” NCT00060996

Remodulin (treprostinil sodium) Injection” NCT00067041

Remodulin (treprostinil sodium)” NCT00494533

NCT02847260

NCT02865733

NCT02261883

NCT01980979

Known as treprostinil diethanolamine “A Randomized, Single-Center, Placebo Controlled Study To Assess the Safety of UT-15C (Treprostinil Diethanolamine) Sustained Release (SR) in Patients Undergoing an...” NCT00651885
4

“A Comparative Bioavailability Study of UT-15C SR (Treprostinil Diethanolamine, Sustained Release) Oral Tablets and UT-15C (Treprostinil Diethanolamine) Administered as an Oral...” NCT01172496

“This study will evaluate the effect of treprostinil diethanolamine (UT-15C) sustained release tablets(compared to placebo) on digital ulcers in patients with scleroderma.” NCT00775463

“Oral UT-15C (Treprostinil Diethanolamine)SR Tablets” NCT00445159

“UT-15C SR (treprostinil diethanolamine)” NCT01131845

Known as treprostinil diolamine “METHODS: We examined 19 circulating vascular, angiogenic, and inflammatory biomarkers in 124 patients with scleroderma and DU who participated in a randomized controlled trial...” PMID 31858338 Dec 2019
1

“UT-15C (treprostinil diolamine)” NCT01560637

Known as treprostinil sodium “Generic treprostinil sodium + Standard of Care (Double Oral)” NCT06317805
8

“Remodulin® (treprostinil sodium) Injection” NCT00060996

“Remodulin (treprostinil sodium) Injection” NCT00067041

“Remodulin (treprostinil sodium)” NCT00494533

“Drug: Treprostinil sodiumNCT01416636

NCT00643604

NCT01884038

NCT00373360

NCT00458042

Known as Tyvaso “Participants will receive inhaled Treprostinil (Tyvaso nebulizer), 6 µg per breath, administered four times daily for 4 weeks.” NCT07037836
2

Tyvaso (treprostinil) inhalation solution” NCT01477333

NCT06193031

Known as Tyvaso DPI “BREEZE: Open-label clinical study to evaluate the safety and tolerability of treprostinil inhalation powder as Tyvaso DPI™ in patients with pulmonary arterial hypertension.” PMID 35514770 Apr 2022
Known as UT-15 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00004497
Known as UT-15C “A Randomized, Single-Center, Placebo Controlled Study To Assess the Safety of UT-15C (Treprostinil Diethanolamine) Sustained Release (SR) in Patients Undergoing an...” NCT00651885
9

“This study is an international, multi-center, open-label study designed to provide oral treprostinil (UT-15C) to eligible subjects with pulmonary arterial hypertension who have...” NCT01560637

“A Comparative Bioavailability Study of UT-15C SR (Treprostinil Diethanolamine, Sustained Release) Oral Tablets and UT-15C (Treprostinil Diethanolamine) Administered as an Oral...” NCT01172496

“This study will evaluate the effect of treprostinil diethanolamine (UT-15C) sustained release tablets(compared to placebo) on digital ulcers in patients with scleroderma.” NCT00775463

“Oral treprostinil (UT-15C), a synthetic prostacyclin analog that inhibits platelet aggregation, induces vasodilation, and suppresses smooth muscle proliferation.” NCT02583789

“randomized (1:1 oral treprostinil (UT-15C): placebo)” NCT01560624

“Oral treprostinil (UT-15C) sustained release tablets” NCT00325442

“Oral treprostinil (UT-15C) Sustained Release Tablets” NCT00325403

“Oral treprostinil (UT-15C) sustained release tablets” NCT07112183

“Oral UT-15C (Treprostinil Diethanolamine)SR Tablets” NCT00445159

Known as UT-15C SR “This study provided/continued to provide oral treprostinil (UT-15C SR; treprostinil diethanolamine) to eligible subjects who participated in Studies TDE-PH-202, TDE-PH-203,...” NCT01027949
2

“A Comparative Bioavailability Study of UT-15C SR (Treprostinil Diethanolamine, Sustained Release) Oral Tablets and UT-15C (Treprostinil Diethanolamine) Administered as an Oral...” NCT01172496

UT-15C SR (treprostinil diethanolamine)” NCT01131845

Known as UT-15C sustained release (SR) “This multi-center, open-label study will assess the tolerability and safety of transitioning subjects with stable Pulmonary Arterial Hypertension (PAH) from continuous...” NCT01588405
Modality Other / unclassified “a prostacyclin analog” NCT00458042
Route Subcutaneous “continuous subcutaneous infusion of either UT-15 or placebo for 12 weeks” NCT00004497