Drugs / Nilutamide
last change Oct 2025 re-read 2 minutes ago

Nilutamide

also known as Anadron · ANAN · Nilandron · Nilutamida · NSC-758683 · RU 23908

Small molecule targets AR

Developed for
prostate cancer
Investigated by
National Cancer Institute (NCI) · M.D. Anderson Cancer Center · SWOG Cancer Research Network

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved US (FDA) NILANDRON 1996-09-19 fda.gov

Trials 3 · a red edge is where a trial was stopped

19961997199819992000200120022003200420052006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 22 trials
Phase 2 NCT00028769 Dec 2001 → Jun 2010 prostate cancer SWOG Cancer Research Network Completed No outcome recorded
Phase 2 NCT00020254 Jun 2000 → Oct 2004 prostate cancer National Cancer Institute (NCI) Completed No outcome recorded
Phase 31 trial
Phase 3 NCT00002855 Aug 1996 → Jun 2005 prostate cancer M.D. Anderson Cancer Center Completed No outcome recorded
Also used as a comparator or background therapy in 9 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT00512668 Background Sep 2007 → Jan 2008 prostate adenocarcinoma National Cancer Institute (NCI) Terminated No outcome recorded
Phase 22 trials
Phase 2 NCT01786265 Background Feb 2013 → Feb 2027 expected prostate adenocarcinoma M.D. Anderson Cancer Center Active not recruiting No outcome recorded
Phase 2 NCT00918385 Comparator May 2009 → Feb 2012 prostate cancer Duke University Terminated No outcome recorded
Phase 2/32 trials
Phase 2/3 NCT04787744 Background Jul 2021 → Sep 2026 expected metastatic prostate carcinoma VA Office of Research and Development Recruiting No outcome recorded
Phase 2/3 NCT03070886 Background Apr 2017 → Oct 2025 prostate adenocarcinoma NRG Oncology Completed No outcome recorded
Phase 34 trials
Phase 3 NCT03678025 Background Sep 2018 → Apr 2028 expected prostate adenocarcinoma SWOG Cancer Research Network Recruiting No outcome recorded
Phase 3 NCT02446405 Comparator Mar 2014 → Dec 2026 expected prostate cancer University of Sydney Active not recruiting No outcome recorded
Phase 3 NCT00003653 Comparator Jan 1999 → Oct 2010 prostate cancer NCIC Clinical Trials Group Completed No outcome recorded
Phase 3 NCT00002633 Comparator Feb 1995 → Sep 2011 prostate cancer NCIC Clinical Trials Group Completed No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 13 sources stand behind the page.

FieldValueCited text
Known as nilutamide “Participants were randomly assigned (1:1), using a centralised web-based system and stratified by volume of disease, planned use of concurrent docetaxel and bone antiresorptive...” PMID 36990608 Apr 2023
11

NCT00003653

NCT03678025

NCT03070886

NCT01786265

NCT00020254

NCT00002855

NCT00002633

NCT04787744

NCT00512668

NCT00918385

NCT00028769

Known as Anadron ChEMBL registry synonym — accepted as the source's own label CHEMBL1274
Known as ANAN “an antiandrogen (nilutamide [ANAN], flutamide [FLUT], bicalutamide [CDX], or cyproterone acetate [CPTR])” NCT00003653
Known as Nilandron ChEMBL registry synonym — accepted as the source's own label CHEMBL1274
Known as Nilutamida ChEMBL registry synonym — accepted as the source's own label CHEMBL1274
Known as NSC-758683 ChEMBL registry synonym — accepted as the source's own label CHEMBL1274
Known as RU 23908 ChEMBL registry synonym — accepted as the source's own label CHEMBL1274
Action Inhibit “Hormone therapy using nilutamide may fight prostate cancer by reducing the production of androgens.” NCT00020254
Modality Small molecule CHEMBL1274
Route Oral “Nilutamide 100 mg po TID x 1 mo; then 150 mg po QD” NCT00002633
Target AR “nilutamide, an approved oral agent used in metastatic CRPC to target the AR.” NCT00918385