Drugs / Lumretuzumab
last change Jan 2018 re-read 2 minutes ago

Lumretuzumab

also known as RO5479599 · RG-7116

Monoclonal antibody targets ERBB3 via inhibition

Developed for
breast cancer · neoplasm · non-small cell squamous lung carcinoma
Investigated by
Hoffmann-La Roche

Trials 3 · a red edge is where a trial was stopped

2012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01918254 Aug 2013 → Oct 2016 breast cancer Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT01482377 Dec 2011 → Feb 2016 neoplasm Hoffmann-La Roche Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT02204345 Oct 2014 → Mar 2016 non-small cell squamous lung carcinoma Hoffmann-La Roche Terminated No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as Lumretuzumab ClinicalTrials.gov intervention name — accepted as the source's own label NCT01918254
Known as RG-7116 ChEMBL registry synonym — accepted as the source's own label CHEMBL3707404
Known as RO5479599 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01482377
1

NCT02204345

Action Inhibit “receptor inhibition using lumretuzumab (anti-HER3) and pertuzumab (anti-HER2)” PMID 29349598 Jan 2018
1

“Receptor tyrosine-protein kinase erbB-3 inhibitor” CHEMBL3707404

Modality Monoclonal antibody CHEMBL3707404
Route Intravenous “Cohorts of participants will receive escalating doses of intravenous RO5479599” NCT01482377
Target ERBB3 “Receptor tyrosine-protein kinase erbB-3 inhibitor” CHEMBL3707404