Drugs / Eluxadoline
last change Apr 2026 re-read 2 minutes ago

Eluxadoline

also known as Eluxadolina · JNJ-27018966 · Truberzi · Viberzi

Small molecule targets OPRM1 via activation

Developed for
irritable bowel syndrome · diarrheal disease · anus disorder · overactive bladder
Investigated by
Allergan · Furiex Pharmaceuticals, Inc · AbbVie · Temple University · University of North Carolina, Chapel Hill

Regulatory milestones approvals, filings & regulatory actions · 3 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Withdrawn EU (EMA) Truberzi 2020-12-18 europa.eu
Approved EU (EMA) Truberzi 2016-09-19 europa.eu
Approved US (FDA) VIBERZI 2015-05-27 fda.gov

Trials 8 · a red edge is where a trial was stopped

201020112012201320142015201620172018201920202021202220232024202520262027202820292030203120322033
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 23 trials
Phase 2 NCT03489265 Apr → Sep 2019 anus disorder, diarrheal disease, overactive bladder University of North Carolina, Chapel Hill Withdrawn No outcome recorded
Phase 2 NCT03339128 Nov 2017 → Dec 2026 expected irritable bowel syndrome AbbVie Recruiting No outcome recorded
Phase 2 NCT01130272 Apr 2010 → Jul 2011 irritable bowel syndrome Furiex Pharmaceuticals, Inc Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT04313088 Jul 2022 → Dec 2023 diabetes mellitus, diarrheal disease Temple University Withdrawn No outcome recorded
Phase 33 trials
Phase 3 NCT04880876 Aug 2021 → Dec 2032 expected irritable bowel syndrome AbbVie Enrolling by invitation No outcome recorded
Phase 3 NCT01553591 May 2012 → Jul 2014 irritable bowel syndrome Furiex Pharmaceuticals, Inc Completed No outcome recorded
Phase 3 NCT01553747 May 2012 → Jan 2014 irritable bowel syndrome Furiex Pharmaceuticals, Inc Completed No outcome recorded
Phase 41 trial
Phase 4 NCT03441581 Feb 2018 → Apr 2020 irritable bowel syndrome Allergan Completed No outcome recorded
Also used as a comparator or background therapy in 2 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 41 trial
Phase 4 NCT02959983 Comparator Oct 2016 → Jan 2018 irritable bowel syndrome Allergan Completed No outcome recorded
Phase not applicable1 trial
NCT07635394 Background Apr 2026 overdue irritable bowel syndrome Beijing Tiantan Hospital Recruiting No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as Eluxadoline Eluxadoline 100 mg BID (75 mg BID in post-cholecystectomy patients)” NCT07635394
9

NCT03441581

NCT04313088

NCT01553591

NCT01553747

NCT03489265

NCT01130272

NCT04880876

NCT02959983

NCT03339128

Known as Eluxadolina ChEMBL registry synonym — accepted as the source's own label CHEMBL2159122
Known as JNJ-27018966 ChEMBL registry synonym — accepted as the source's own label CHEMBL2159122
Known as Truberzi ChEMBL registry synonym — accepted as the source's own label CHEMBL2159122
Known as Viberzi ChEMBL registry synonym — accepted as the source's own label CHEMBL2159122
Action Activate “Mu opioid receptor agonist” CHEMBL2159122
Modality Small molecule CHEMBL2159122
Route Oral “5, 25, 100, or 200 mg oral eluxadoline” PMID 23583433 Apr 2013
Target OPRM1 “Mu opioid receptor agonist” CHEMBL2159122