Drugs / Evofosfamide
last change May 2026 re-read 2 minutes ago

Evofosfamide

Other / unclassified

Developed for
malignant pancreatic neoplasm · soft tissue sarcoma · cancer · head and neck squamous cell carcinoma · non-small cell lung carcinoma · pancreatic adenocarcinoma · prostate cancer · acute myeloid leukemia
+21 more · biliary tract cancer · castration-resistant prostate carcinoma · chronic lymphocytic leukemia/small lymphocytic lymphoma · chronic myeloid leukemia · esophageal cancer · gastrointestinal stromal tumor · glioblastoma · hepatocellular carcinoma · high grade astrocytic tumor · kidney cancer · liver cancer · melanoma · metastatic melanoma · metastatic prostate carcinoma · myelodysplastic syndrome · myelofibrosis · neoplasm · pancreatic neuroendocrine neoplasm · pancreatic neuroendocrine tumor · plasma cell myeloma · renal cell carcinoma
Investigated by
Threshold Pharmaceuticals · ImmunoGenesis · Merck KGaA, Darmstadt, Germany · Sarcoma Alliance for Research through Collaboration · The University of Texas Health Science Center at San Antonio · Agenus Inc.
+15 more · Alliance for Clinical Trials in Oncology · EMD Serono · GlaxoSmithKline · Herbert Hurwitz, MD · M.D. Anderson Cancer Center · Maastricht Radiation Oncology · National Cancer Institute (NCI) · National Comprehensive Cancer Network · PRA Health Sciences · Pfizer · Scripps Clinic Cancer Center · Seoul National University Hospital · Spanish Group for Research in Neuroendocrine Tumors · University Health Network, Toronto · Zuyderland Medical Centre

Trials 27 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 112 trials
Phase 1 NCT03098160 May 2017 → Jan 2019 head and neck squamous cell carcinoma, malignant pancreatic neoplasm, melanoma, prostate cancer Threshold Pharmaceuticals Unknown No outcome recorded
Phase 1 NCT02598687 Dec 2015 → Apr 2016 esophageal cancer Maastricht Radiation Oncology Withdrawn No outcome recorded
Phase 1 NCT01721941 Dec 2014 → Dec 2015 hepatocellular carcinoma Scripps Clinic Cancer Center Unknown No outcome recorded
Phase 1 NCT02076230 Feb → Sep 2014 cancer Merck KGaA, Darmstadt, Germany Completed No outcome recorded
Phase 1 NCT02047500 Jan 2014 → Sep 2015 pancreatic adenocarcinoma ImmunoGenesis Terminated No outcome recorded
Phase 1 NCT02020226 Nov 2013 → Jul 2016 cancer Threshold Pharmaceuticals Unknown No outcome recorded
Phase 1 NCT01833546 Apr 2013 → Aug 2015 malignant pancreatic neoplasm Merck KGaA, Darmstadt, Germany Completed No outcome recorded
Phase 1 NCT01497444 May 2012 → Jan 2016 kidney cancer, liver cancer Alliance for Clinical Trials in Oncology Completed No outcome recorded
Phase 1 NCT01485042 Dec 2011 → Feb 2013 cancer Herbert Hurwitz, MD Completed No outcome recorded
Phase 1 NCT01381822 Jun 2011 → Jun 2014 gastrointestinal stromal tumor, pancreatic neuroendocrine tumor, renal cell carcinoma Threshold Pharmaceuticals Unknown No outcome recorded
Phase 1/24 trials
Phase 1/2 NCT06782555 Jan 2025 → Oct 2027 expected head and neck squamous cell carcinoma, malignant pancreatic neoplasm, metastatic prostate carcinoma ImmunoGenesis Recruiting No outcome recorded
Phase 1/2 NCT01522872 Feb 2012 → Sep 2016 plasma cell myeloma Threshold Pharmaceuticals Unknown No outcome recorded
Phase 1/2 NCT00742963 Aug 2008 → Jul 2013 soft tissue sarcoma ImmunoGenesis Completed No outcome recorded
Phase 1/2 NCT00743379 Aug 2008 → Jul 2013 malignant pancreatic neoplasm, non-small cell lung carcinoma, prostate cancer Threshold Pharmaceuticals Completed No outcome recorded
Phase 29 trials
Phase 2 NCT06836726 May 2026 → May 2028 expected castration-resistant prostate carcinoma University Health Network, Toronto Not yet recruiting No outcome recorded
Phase 2 NCT02402062 May 2015 → May 2018 pancreatic neuroendocrine neoplasm Spanish Group for Research in Neuroendocrine Tumors Completed No outcome recorded
Phase 2 NCT02342379 May 2015 → Jan 2019 glioblastoma The University of Texas Health Science Center at San Antonio Completed No outcome recorded
Phase 2 NCT02433639 Apr 2015 → Oct 2017 biliary tract cancer Seoul National University Hospital Completed No outcome recorded
Phase 2 NCT02255110 Dec 2014 → Jan 2016 soft tissue sarcoma Merck KGaA, Darmstadt, Germany Terminated No outcome recorded
Phase 2 NCT02093962 Jun 2014 → Apr 2016 non-small cell lung carcinoma ImmunoGenesis Terminated No outcome recorded
Phase 2 NCT01864538 May 2013 → Sep 2015 metastatic melanoma ImmunoGenesis Terminated No outcome recorded
Phase 2 NCT01403610 Jun 2011 → Oct 2015 high grade astrocytic tumor The University of Texas Health Science Center at San Antonio Completed No outcome recorded
Phase 2 NCT01144455 Jun 2010 → Sep 2013 pancreatic adenocarcinoma ImmunoGenesis Completed No outcome recorded
Phase 31 trial
Phase 3 NCT01440088 Sep 2011 → Dec 2015 soft tissue sarcoma Threshold Pharmaceuticals Completed No outcome recorded
Phase not stated1 trial
NCT02712567 soft tissue sarcoma Sarcoma Alliance for Research through Collaboration No longer available No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 3 NCT01746979 Comparator Dec 2012 → Feb 2016 pancreatic adenocarcinoma ImmunoGenesis Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 32 sources stand behind the page.

FieldValueCited text
Known as evofosfamide “A phase 1 'window-of-opportunity' trial testing evofosfamide (TH-302), a tumour-selective hypoxia-activated cytotoxic prodrug, with preoperative chemoradiotherapy in...” PMID 27535748 Aug 2016
5

“Sunitinib and Evofosfamide (TH-302) in Systemic Treatment-naïve Patients with Grade 1/2 Metastatic Pancreatic Neuroendocrine Tumors: The GETNE-1408 Trial.” PMID 34190375 Jul 2021

NCT06782555

NCT06836726

NCT03098160

NCT01833546

Known as EVO “Sunitinib and Evofosfamide (TH-302) in Systemic Treatment-naïve Patients with Grade 1/2 Metastatic Pancreatic Neuroendocrine Tumors: The GETNE-1408 Trial.” PMID 34190375 Jul 2021
Known as Evofosfamida ChEMBL registry synonym — accepted as the source's own label CHEMBL260046
Known as HAP-302 ChEMBL registry synonym — accepted as the source's own label CHEMBL260046
Known as TH-302 “The goal of this study is to provide continuation therapy with TH-302 to patients with soft tissue sarcomas who obtained response or stabilization of disease with prior...” NCT02712567
24

“The dose of TH-302 will be mixed with doxorubicin 50mg to use as the chemoembolization mixture for transarterial chemoembolization (TACE).” NCT01721941

NCT00495144

NCT00742963

NCT01485042

NCT01746979

NCT00743379

NCT02712567

NCT02402062

NCT01497444

NCT02433639

NCT02020226

NCT01144455

NCT02342379

NCT01864538

NCT02093962

NCT01381822

NCT01522872

NCT02076230

NCT01440088

NCT02255110

NCT01403610

NCT02047500

NCT01149915

NCT02598687

Known as TH-302 (1-methyl-2-nitro-1H-imidazole-5-yl)methyl N,N'-bis(2-bromoethyl) diamidophos-phate TH-302 (1-methyl-2-nitro-1H-imidazole-5-yl)methyl N,N'-bis(2-bromoethyl) diamidophos-phate is a nitroimidazole-linked prodrug of a brominated version of isophosphoramide...” NCT02433639
Modality Other / unclassified “TH-302 is an investigational hypoxia-activated prodrug” PMID 25512461 Dec 2014
Route Intravenous “TH-302 will be administered by IV infusion over 30-60 minutes” NCT00742963