Drugs / AZD2066
last change Nov 2010 re-read 9 days ago

AZD2066

Small molecule targets GRM5

Developed for
diabetic neuropathy · major depressive disorder · myofascial pain syndrome · neuropathy, painful
Investigated by
AstraZeneca · Quintiles, Inc.

Trials 10

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT00930306 Jun → Sep 2009 chronic pain syndrome AstraZeneca Completed No outcome recorded
Phase 1 NCT00829088 Jan → Feb 2009 — AstraZeneca Completed No outcome recorded
Phase 1 NCT00766012 Sep 2008 → Jul 2009 — AstraZeneca Completed No outcome recorded
Phase 1 NCT00686504 Apr → Jun 2008 — AstraZeneca Completed No outcome recorded
Phase 1 NCT00690404 Apr → Jun 2008 — AstraZeneca Completed No outcome recorded
Phase 1 NCT00684502 Jan → Nov 2008 — AstraZeneca Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00813306 Dec 2008 → Nov 2009 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 23 trials
Phase 2 NCT01145755 May → Nov 2010 major depressive disorder AstraZeneca Terminated No outcome recorded
Phase 2 NCT00939094 Aug 2009 → Nov 2010 myofascial pain syndrome, neuropathy, painful AstraZeneca Terminated No outcome recorded
Phase 2 NCT00857623 Feb → Aug 2009 diabetic neuropathy AstraZeneca Completed No outcome recorded

Evidence & citations 4 cited values

Every value below carries the sentence it was read from. 11 sources stand behind the page.

FieldValueCited text
Known as AZD2066 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01145755 ↗
9

NCT00690404 ↗

NCT00930306 ↗

NCT00857623 ↗

NCT00939094 ↗

NCT00813306 ↗

NCT00829088 ↗

NCT00686504 ↗

NCT00684502 ↗

NCT00766012 ↗

Modality Small molecule — CHEMBL3545164 ↗
Route Oral “Oral solution administered orally once per day on day 1, and then day 3 through to day 12.” NCT00684502 ↗
Target GRM5 “Metabotropic glutamate receptor 5 modulator” CHEMBL3545164 ↗