Drugs / EDELINONTRINE
last change Jul 2023 re-read 2 minutes ago

EDELINONTRINE

also known as PF-04447943 · CRD-740 · Edelinontrina · PF-4447943

Small molecule targets PDE9A via inhibition

Developed for
Alzheimer disease · sickle cell disease · symptomatic heart failure
Investigated by
Pfizer · Cardurion Pharmaceuticals, Inc.

Trials 10 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 18 trials
Phase 1 NCT05437094 Jun → Aug 2022 heart failure Cardurion Pharmaceuticals, Inc. Completed No outcome recorded
Phase 1 NCT02785770 Jun → Oct 2016 Pfizer Completed No outcome recorded
Phase 1 NCT02114203 Dec 2014 → Sep 2016 sickle cell disease Pfizer Completed No outcome recorded
Phase 1 NCT01097876 Apr → Jul 2010 Pfizer Completed No outcome recorded
Phase 1 NCT00959803 Aug → Nov 2009 Pfizer Completed No outcome recorded
Phase 1 NCT00886093 Apr → May 2009 Pfizer Completed No outcome recorded
Phase 1 NCT00832052 Jan → May 2009 Pfizer Completed No outcome recorded
Phase 1 NCT00736528 Aug → Sep 2008 Pfizer Terminated No outcome recorded
Phase 22 trials
Phase 2 NCT05409183 May 2022 → May 2023 symptomatic heart failure Cardurion Pharmaceuticals, Inc. Terminated No outcome recorded
Phase 2 NCT00930059 Sep 2009 → Sep 2010 Alzheimer disease Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT00988598 Comparator Oct 2009 → Jul 2010 Alzheimer disease Pfizer Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as EDELINONTRINE ChEMBL registry synonym — accepted as the source's own label CHEMBL2179105
Known as CRD-740 ClinicalTrials.gov intervention name — accepted as the source's own label NCT05409183
1

NCT05437094

Known as Edelinontrina ChEMBL registry synonym — accepted as the source's own label CHEMBL2179105
Known as PF-04447943 PF-04447943, a Phosphodiesterase 9A Inhibitor, in Stable Sickle Cell Disease” PMID 30597771 Dec 2018
8

NCT01097876

NCT00930059

NCT00886093

NCT00736528

NCT00988598

NCT00832052

NCT00959803

NCT02785770

Known as PF-4447943 ChEMBL registry synonym — accepted as the source's own label CHEMBL2179105
Action Inhibit “PF-04447943, a phosphodiesterase 9A inhibitor” PMID 30597771 Dec 2018
Modality Small molecule CHEMBL2179105
Route Oral “multiple, ascending, oral doses” NCT00736528
Target PDE9A “PF-04447943, a phosphodiesterase 9A inhibitor” PMID 30597771 Dec 2018