Drugs / ZIMLOVISERTIB
last change May 2022 re-read 2 minutes ago

ZIMLOVISERTIB

Small molecule targets IRAK4 via inhibition

Developed for
rheumatoid arthritis · COVID-19 · hidradenitis suppurativa · pneumonia
Investigated by
Pfizer · Yale University

Trials 11 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 17 trials
Phase 1 NCT05064332 Oct → Dec 2021 Pfizer Completed No outcome recorded
Phase 1 NCT03827668 Feb → Apr 2019 Pfizer Completed No outcome recorded
Phase 1 NCT03308110 Sep → Dec 2017 Pfizer Completed No outcome recorded
Phase 1 NCT02936154 Aug → Oct 2016 Pfizer Completed No outcome recorded
Phase 1 NCT02609139 Nov 2015 → Feb 2016 Pfizer Completed No outcome recorded
Phase 1 NCT02485769 Jun 2015 → Apr 2016 Pfizer Completed No outcome recorded
Phase 1 NCT02224651 Sep 2014 → Jun 2015 Pfizer Completed No outcome recorded
Phase 24 trials
Phase 2 NCT04575610 Nov 2020 → Oct 2021 COVID-19 Yale University Terminated No outcome recorded
Phase 2 NCT04413617 Jul 2020 → Feb 2022 rheumatoid arthritis Pfizer Completed No outcome recorded
Phase 2 NCT04092452 Dec 2019 → Jan 2022 hidradenitis suppurativa Pfizer Completed No outcome recorded
Phase 2 NCT02996500 Nov 2016 → Aug 2018 rheumatoid arthritis Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT04933799 Comparator Jan 2021 → Mar 2022 pneumonia Giovanni Franchin, M.D, Ph.D Unknown No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 15 sources stand behind the page.

FieldValueCited text
Known as ZIMLOVISERTIB ChEMBL registry synonym — accepted as the source's own label CHEMBL4081711
Known as PF-06650833 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02936154
11

NCT03308110

NCT04933799

NCT04092452

NCT04413617

NCT03827668

NCT02609139

NCT02224651

NCT04575610

NCT02996500

NCT05064332

NCT02485769

Known as ZIMLOVISERTIB (PF-06650833) ChEMBL registry synonym — accepted as the source's own label CHEMBL4081711
Action Inhibit “PF-06650833 is a potent, selective inhibitor of interleukin-1 receptor-associated kinase 4 (IRAK4).” PMID 31805989 Dec 2019
Modality Small molecule “a highly potent and selective small-molecule inhibitor of interleukin-1-associated kinase 4 (IRAK4)” PMID 34423919 Nov 2021
Route Oral oral PF-06650833 IR 1 to 6000 mg” PMID 31805989 Dec 2019
Target IRAK4 “PF-06650833 is a potent, selective inhibitor of interleukin-1 receptor-associated kinase 4 (IRAK4).” PMID 31805989 Dec 2019