Drugs / PF-03654746
last change Apr 2012 re-read 2 minutes ago

PF-03654746

Small molecule targets HRH3 via inhibition

Developed for
allergic rhinitis · Alzheimer disease · attention deficit-hyperactivity disorder · hypersomnia · narcolepsy · schizophrenia · Tourette syndrome
Investigated by
Pfizer · Yale University

Trials 4 · a red edge is where a trial was stopped

20082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01028911 Dec 2009 → May 2010 Alzheimer disease Pfizer Terminated No outcome recorded
Phase 1 NCT00730990 May → Nov 2008 Pfizer Completed No outcome recorded
Phase 22 trials
Phase 2 NCT00531752 Dec 2007 → Sep 2008 attention deficit-hyperactivity disorder Pfizer Completed No outcome recorded
Phase 2 NCT00562120 Dec 2007 → Aug 2008 allergic rhinitis Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 3 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT01346163 Comparator Apr 2009 → Nov 2010 schizophrenia University of Pennsylvania Completed No outcome recorded
Phase 22 trials
Phase 2 NCT01475383 Comparator Apr 2012 Tourette syndrome Pfizer Withdrawn No outcome recorded
Phase 2 NCT01006122 Comparator Nov 2009 → Nov 2010 hypersomnia, narcolepsy Pfizer Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as PF 03654746 “This study will look at the impact of dosing as well as ongoing treatment with an investigation medication identified as PF-03654746, on cognitive and physiologic indicators of...” NCT01346163
7

“Drug: PF 03654746NCT01346163

NCT00730990

NCT01028911

NCT01475383

NCT00562120

NCT00531752

NCT01006122

Action Inhibit “Histamine H3 receptor antagonist” CHEMBL2151197
1

“H3 receptor antagonist” NCT01346163

Modality Small molecule CHEMBL2151197
Route Oral “A single oral dose of PF-03654746 is the investigational drug being studied.” NCT00562120
Target HRH3 “Histamine H3 receptor antagonist” CHEMBL2151197