Drugs / TS-142
last change Mar 2024 re-read 2 minutes ago

TS-142

English name vornorexant
also known as vornorexant

Small molecule

Developed for
insomnia · obstructive sleep apnea syndrome
Investigated by
Taisho Pharmaceutical Co., Ltd. · Taisho Pharmaceutical R&D Inc.

Trials 15 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 111 trials
Phase 1 NCT05819710 May → Aug 2023 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT05707897 Feb → Mar 2023 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT05624944 Dec 2022 → Dec 2023 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT04873323 Jun → Sep 2021 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT04814771 Apr → May 2021 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT04746105 Feb → Oct 2021 obstructive sleep apnea syndrome Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT04696952 Jan 2021 → Jan 2022 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT04557163 Oct → Nov 2020 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT04464239 Sep 2020 → Jan 2021 Taisho Pharmaceutical R&D Inc. Completed No outcome recorded
Phase 1 NCT04169906 Jul → Oct 2016 Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 22 trials
Phase 2 NCT04469023 Sep 2020 → Nov 2021 insomnia Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 2 NCT04573725 Jul 2017 → Feb 2019 insomnia Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 32 trials
Phase 3 NCT05461352 Oct 2022 → Mar 2024 insomnia Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 3 NCT05453136 Aug 2022 → Dec 2023 insomnia Taisho Pharmaceutical Co., Ltd. Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 17 sources stand behind the page.

FieldValueCited text
Known as TS-142 ClinicalTrials.gov intervention name — accepted as the source's own label NCT04169893
14

NCT05453136

NCT04464239

NCT05461352

NCT05624944

NCT04557163

NCT04873323

NCT04696952

NCT04746105

NCT04469023

NCT05819710

NCT05707897

NCT04169906

NCT04814771

NCT04573725

Known as vornorexant “receptor antagonist vornorexant/TS-142 in healthy Japanese participants” PMID 37563858 Sep 2023
Action Inhibit “dual orexin receptor antagonist” PMID 37563858 Sep 2023
Modality Small molecule “Novel compound with potent antagonistic activity against orexin receptors may be new treatment option for patients with insomnia.” PMID 35296912 Mar 2022
Route Oral “single oral doses” NCT04464239