Drugs / Padsevonil
last change Jul 2024 re-read 2 minutes ago

Padsevonil

also known as UCB0942 · PSL · UCB-1415943-000

Small molecule targets CYP2C19, CYP3A4

Developed for
focal epilepsy
Investigated by
UCB Biopharma S.P.R.L. · UCB Biopharma SRL · PRA Health Sciences

Trials 14 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 19 trials
Phase 1 NCT04136444 Oct 2019 → May 2020 UCB Biopharma S.P.R.L. Terminated No outcome recorded
Phase 1 NCT04126343 Oct 2019 → May 2020 UCB Biopharma S.P.R.L. Terminated No outcome recorded
Phase 1 NCT04131517 Oct 2019 → May 2020 UCB Biopharma SRL Terminated No outcome recorded
Phase 1 NCT04075409 Sep → Dec 2019 UCB Biopharma S.P.R.L. Completed No outcome recorded
Phase 1 NCT04039919 Jul 2019 → May 2020 UCB Biopharma S.P.R.L. Terminated No outcome recorded
Phase 1 NCT04013191 Jul → Oct 2019 UCB Biopharma S.P.R.L. Completed No outcome recorded
Phase 1 NCT03695094 Sep 2018 → May 2019 epilepsy UCB Biopharma S.P.R.L. Completed No outcome recorded
Phase 1 NCT03480243 Mar → Aug 2018 UCB Biopharma S.P.R.L. Completed No outcome recorded
Phase 1 NCT03168984 May → Aug 2017 UCB Biopharma S.P.R.L. Completed No outcome recorded
Phase 24 trials
Phase 2 NCT03370120 Aug 2018 → Dec 2020 focal epilepsy UCB Biopharma SRL Terminated No outcome recorded
Phase 2 NCT03373383 Feb 2018 → Jan 2020 focal epilepsy UCB Biopharma S.P.R.L. Completed No outcome recorded
Phase 2 NCT02625090 Dec 2015 → Nov 2020 focal epilepsy UCB Biopharma SRL Terminated No outcome recorded
Phase 2 NCT02495844 Jul 2015 → Feb 2017 focal epilepsy UCB Biopharma S.P.R.L. Completed No outcome recorded
Phase 31 trial
Phase 3 NCT03739840 Mar 2019 → Sep 2020 focal epilepsy UCB Biopharma SRL Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT04283136 Comparator Feb → May 2020 epilepsy UCB Biopharma SRL Withdrawn No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 18 sources stand behind the page.

FieldValueCited text
Known as Padsevonil ClinicalTrials.gov intervention name — accepted as the source's own label NCT04136444
11

NCT03370120

NCT04013191

NCT03739840

NCT03373383

NCT03695094

NCT04075409

NCT04131517

NCT03480243

NCT04039919

NCT04283136

NCT04126343

Known as PSL “The purpose of the study in Part 1, is to evaluate (under fasted conditions) the plasma pharmacokinetics (PK) of padsevonil (PSL) using 4 PSL product variants against a PSL...” NCT04283136
2

“To characterize efficacy, safety/tolerability, and pharmacokinetics of padsevonil (PSL) administered concomitantly with ≤3 antiseizure medications (ASMs) for observable focal...” PMID 36176044 Oct 2022

“The purpose of the study is to evaluate the pharmacodynamic (PD) interaction between steady-steady treatment with padsevonil (PSL) and Ethanol and the pharmacokinetic (PK)...” NCT04039919

Known as UCB-1415943-000 ChEMBL registry synonym — accepted as the source's own label CHEMBL4297521
Known as UCB0942 “Padsevonil (UCB0942)” NCT03480243
3

NCT02495844

NCT03168984

NCT02625090

Modality Small molecule CHEMBL4297521
Route Oral “Route of Administration: Oral use” NCT02495844
Target CYP2C19 “Padsevonil was shown to be a time-dependent CYP2C19-inhibitor, weak CYP3A4-inducer, weak inhibitor of P-gp/OCT1/MATE2-K, and potent OCT2-inhibitor.” PMID 38932723 Jul 2024
Target CYP3A4 “Padsevonil was shown to be a time-dependent CYP2C19-inhibitor, weak CYP3A4-inducer, weak inhibitor of P-gp/OCT1/MATE2-K, and potent OCT2-inhibitor.” PMID 38932723 Jul 2024