Drugs / PEGPLERANIB SODIUM
last change Jul 2019 re-read 2 minutes ago

PEGPLERANIB SODIUM

also known as E10030 · Fovista · E-01AJ · X-01E

Aptamer targets PDGFB via inhibition

Developed for
age-related macular degeneration · von Hippel-Lindau disease · wet macular degeneration
Investigated by
Ophthotech Corporation · National Eye Institute (NEI) · Retinal Consultants of Arizona

Trials 8 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT02591914 Feb 2014 → May 2016 wet macular degeneration Retinal Consultants of Arizona Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT02859441 Jan 2017 → Jul 2019 von Hippel-Lindau disease National Eye Institute (NEI) Completed No outcome recorded
Phase 23 trials
Phase 2 NCT02387957 Apr 2016 → Jan 2017 age-related macular degeneration Ophthotech Corporation Terminated No outcome recorded
Phase 2 NCT02214628 Jul 2014 → Dec 2016 age-related macular degeneration Ophthotech Corporation Terminated No outcome recorded
Phase 2 NCT01089517 Mar 2010 → Jun 2012 age-related macular degeneration Ophthotech Corporation Completed No outcome recorded
Phase 33 trials
Phase 3 NCT01940887 May 2014 → Jun 2017 age-related macular degeneration Ophthotech Corporation Terminated No outcome recorded
Phase 3 NCT01944839 Aug 2013 → Dec 2016 age-related macular degeneration Ophthotech Corporation Terminated No outcome recorded
Phase 3 NCT01940900 Aug 2013 → Dec 2016 age-related macular degeneration Ophthotech Corporation Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT00569140 Comparator Dec 2007 → Dec 2008 age-related macular degeneration Ophthotech Corporation Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 10 sources stand behind the page.

FieldValueCited text
Known as PEGPLERANIB SODIUM ChEMBL registry synonym — accepted as the source's own label CHEMBL3301576
Known as E-01AJ ChEMBL registry synonym — accepted as the source's own label CHEMBL3301576
Known as E10030 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01940887
5

NCT01944839

NCT02859441

NCT01089517

NCT01940900

NCT00569140

Known as Fovista “A Phase 3 Safety and Efficacy Study of Fovista® (E10030) Intravitreous Administration in Combination With Lucentis® Compared to Lucentis® Monotherapy” NCT01944839
3

NCT02214628

NCT02591914

NCT02387957

Known as X-01E ChEMBL registry synonym — accepted as the source's own label CHEMBL3301576
Action Inhibit “Anti-PDGF” NCT00569140
Modality Aptamer “Anti-PDGF Pegylated AptamerNCT00569140
Route Intravitreal Intravitreal injection” NCT00569140
Target PDGFB “Anti PDGF-B Pegylated Aptamer” NCT01944839