Drugs / PF-05089771
last change Sep 2023 re-read 2 minutes ago

PF-05089771

Small molecule targets SCN9A via inhibition

Developed for
diabetic polyneuropathy · primary erythermalgia
Investigated by
Pfizer · Medical University of Vienna

Trials 13 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT05935280 Jul → Sep 2023 Medical University of Vienna Completed No outcome recorded
Phase 19 trials
Phase 1 NCT02349607 Jan → Mar 2015 Pfizer Completed No outcome recorded
Phase 1 NCT01934569 Sep → Nov 2013 Pfizer Completed No outcome recorded
Phase 1 NCT01854996 May → Jun 2013 Pfizer Completed No outcome recorded
Phase 1 NCT01772264 Jan → Apr 2013 Pfizer Completed No outcome recorded
Phase 1 NCT01690351 Sep 2012 Pfizer Completed No outcome recorded
Phase 1 NCT01563497 Feb 2012 Pfizer Completed No outcome recorded
Phase 1 NCT01529671 Jan → Oct 2012 Pfizer Completed No outcome recorded
Phase 1 NCT01365637 Jun → Sep 2011 Pfizer Completed No outcome recorded
Phase 1 NCT01259882 Dec 2010 → Sep 2011 Pfizer Completed No outcome recorded
Phase 23 trials
Phase 2 NCT02215252 Nov 2014 → Jul 2015 diabetic polyneuropathy Pfizer Completed No outcome recorded
Phase 2 NCT01769274 Oct 2012 → Jul 2013 primary erythermalgia Pfizer Completed No outcome recorded
Phase 2 NCT01529346 Dec 2011 → Jun 2012 Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT01165736 Comparator Jul → Aug 2010 Pfizer Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 16 sources stand behind the page.

FieldValueCited text
Known as PF-05089771 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01934569
13

NCT01690351

NCT01529346

NCT01854996

NCT01365637

NCT01259882

NCT02215252

NCT01772264

NCT01165736

NCT01769274

NCT01529671

NCT02349607

NCT05935280

NCT01563497

Action Inhibit “Sodium channel protein type IX alpha subunit blocker” CHEMBL2325014
1

“blocked the Nav1.7 sodium channel” PMID 27099175 Apr 2016

Modality Small molecule “treated with a new potent and selective compound that blocked the Nav1.7 sodium channel” PMID 27099175 Apr 2016
Route Intravenous “single intravenous infusion of 100 microgram of PF-05089771” NCT01165736
Target SCN9A “Sodium channel protein type IX alpha subunit blocker” CHEMBL2325014