Drugs / Icaritin
last change Jun 2026 re-read 2 minutes ago

Icaritin

also known as Icaritin soft capsule · SGN-162

Small molecule targets TNF via inhibition

Developed for
hepatocellular carcinoma · breast cancer · cancer · colorectal cancer · pancreatic ductal adenocarcinoma
Investigated by
Beijing Shenogen Biomedical Co., Ltd · Chinese Academy of Medical Sciences · 307 Hospital of PLA · Affiliated Cancer Hospital & Institute of Guangzhou Medical University · Anhui Provincial Hospital · Beijing Hospital
+45 more · First People's Hospital of Foshan · Fudan University · Guang'anmen Hospital of China Academy of Chinese Medical Sciences · Hebei Medical University Fourth Hospital · Henan Cancer Hospital · Jinan Central Hospital · NanJing PLA 81 Hospital · Nanfang Hospital, Southern Medical University · Peking University Cancer Hospital & Institute · Sir Run Run Shaw Hospital · The Affiliated Tumor Hospital of Nantong University, Nantong, Jiangsu Province, China · The First Affiliated Hospital of Anhui Medical University · The First Affiliated Hospital with Nanjing Medical University · The First Hospital of Jilin University · Beijing YouAn Hospital · Cancer Institute and Hospital, Chinese Academy of Medical Sciences · Chifeng Municipal Hospital · Chinese PLA General Hospital · Chongqing Traditional Chinese Medicine Hospital · Eastern Theater General Hospital,QinHuai District Medical Area · First Affiliated Hospital of Harbin Medical University · General Hospital of Chinese Armed Police Forces · Guilin Medical University, China · Haikou People's Hospital · Hangzhou Zhongmei Huadong Pharmaceutical Co., Ltd. · Hunan Cancer Hospital · Jilin Provincial Tumor Hospital · Linyi Cancer Hospital · Linyi Tumour Hospital · Nanjing Tianyinshan Hospital · Northern Jiangsu People's Hospital · Qingdao University · Second Affiliated Hospital, School of Medicine, Zhejiang University · Shenyang Sixth People's Hospital · The Affiliated Hospital of Hangzhou Normal University · The First Affiliated Hospital of Bengbu Medical University · The First Affiliated Hospital of Soochow University · The First Affiliated Hospital of Zhengzhou University · The Third Xiangya Hospital of Central South University · Tianjin Medical University Cancer Institute and Hospital · Tongji Hospital · West China Hospital · Yunnan Provincial Hospital of Traditional Chinese Medicine · Zhejiang Cancer Hospital · Zhiyong Huang

Trials 14 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT02496949 Nov 2011 → May 2013 cancer Chinese Academy of Medical Sciences Completed No outcome recorded
Phase 1 NCT01278810 Nov 2010 → Nov 2011 breast cancer Chinese Academy of Medical Sciences Unknown No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT06896396 Apr 2025 → Jun 2027 expected hepatocellular carcinoma Zhiyong Huang Not yet recruiting No outcome recorded
Phase 26 trials
Phase 2 NCT07337460 Nov 2025 → Nov 2027 expected hepatocellular carcinoma Northern Jiangsu People's Hospital Recruiting No outcome recorded
Phase 2 NCT06825546 Apr 2025 → Apr 2027 expected pancreatic ductal adenocarcinoma Sir Run Run Shaw Hospital Recruiting No outcome recorded
Phase 2 NCT06285149 Mar → Dec 2024 hepatocellular carcinoma Henan Cancer Hospital Unknown No outcome recorded
Phase 2 NCT07328828 Mar 2024 → Mar 2025 overdue Second Affiliated Hospital, School of Medicine, Zhejiang University Active not recruiting No outcome recorded
Phase 2 NCT05903456 Jul 2023 → May 2025 hepatocellular carcinoma Zhejiang Cancer Hospital Unknown No outcome recorded
Phase 2 NCT01972672 Oct 2013 → Aug 2015 hepatocellular carcinoma Beijing Shenogen Biomedical Co., Ltd Completed No outcome recorded
Phase 33 trials
Phase 3 NCT05594927 Dec 2022 → Aug 2025 overdue hepatocellular carcinoma Beijing Shenogen Biomedical Co., Ltd Recruiting No outcome recorded
Phase 3 NCT03236649 Sep 2017 → Feb 2022 hepatocellular carcinoma Beijing Shenogen Biomedical Co., Ltd Terminated No outcome recorded
Phase 3 NCT03236636 Sep 2017 → Dec 2022 hepatocellular carcinoma Beijing Shenogen Biomedical Co., Ltd Unknown No outcome recorded
Phase 41 trial
Phase 4 NCT06269445 Jan 2024 → Feb 2025 colorectal cancer Sir Run Run Shaw Hospital Unknown No outcome recorded
Phase not applicable1 trial
NCT06893887 May 2025 → Mar 2027 expected hepatocellular carcinoma Nanjing Tianyinshan Hospital Recruiting No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 15 sources stand behind the page.

FieldValueCited text
Known as Icaritin ClinicalTrials.gov intervention name — accepted as the source's own label NCT03236636
13

NCT07328828

NCT06893887

NCT01278810

NCT05903456

NCT07337460

NCT01972672

NCT06285149

NCT06896396

NCT06269445

NCT02496949

NCT05594927

NCT06825546

NCT03236649

Known as Icaritin soft capsule Icaritin soft capsule is a flavonoid compound extracted from traditional Chinese medicinal materials.” NCT05903456
Known as SGN-162 ChEMBL registry synonym — accepted as the source's own label CHEMBL498485
Action Inhibit “By inhibiting inflammatory signaling pathway and reducing the release of inflammatory factors, the immune microenvironment can be regulated to play an anti-tumor role.” NCT05903456
Modality Small molecule “Icaritin is a newly discovered small molecular compound” NCT01278810
Route Oral “ascending-multiple oral dose” NCT01278810
Target TNF “Icaritin can downregulate the expression of TNF-α, IL-6, PD-L1” NCT06285149