Drugs / Xenin-25
last change Jul 2018 re-read 2 minutes ago

Xenin-25

also known as Xen

Peptide targets NTSR1 via activation

Developed for
diabetes mellitus · type 2 diabetes mellitus
Investigated by
Washington University School of Medicine · National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK) · American Diabetes Association

Trials 5 · a red edge is where a trial was stopped

2009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT02204813 Jul 2014 → Nov 2015 Washington University School of Medicine Completed No outcome recorded
Phase 1 NCT01951729 Mar 2013 → May 2015 prediabetes syndrome Washington University School of Medicine Completed No outcome recorded
Phase 1 NCT01951716 Jan 2013 → Jul 2018 Washington University School of Medicine Withdrawn No outcome recorded
Phase 1 NCT00949663 Oct 2009 → Feb 2014 type 2 diabetes mellitus Washington University School of Medicine Completed No outcome recorded
Phase 1 NCT00798915 Dec 2008 → Dec 2012 diabetes mellitus Washington University School of Medicine Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as Xenin-25 Xenin-25 (Xen) is a neurotensin-related peptide secreted by a subset of enteroendocrine cells located in the proximal small intestine.” PMID 27288245 Jun 2016
4

NCT00798915

NCT01951716

NCT01951729

NCT00949663

Known as Xen Xenin-25 (Xen) is a neurotensin-related peptide secreted by a subset of glucose-dependent insulinotropic polypeptide (GIP)-producing enteroendocrine cells.” PMID 24356886 Dec 2013
2

Xenin-25 (Xen) is a neurotensin-related peptide secreted by a subset of enteroendocrine cells located in the proximal small intestine.” PMID 27288245 Jun 2016

Xenin-25 (Xen) is a 25-amino acid neurotensin-related peptide that activates neurotensin receptor-1 (NTSR1).” PMID 24183983 Oct 2013

Action Activate activates neurotensin receptor-1 (NTSR1)” PMID 24183983 Oct 2013
Modality Peptide “Xenin-25 (Xen) is a 25-amino acid neurotensin-related peptidePMID 24183983 Oct 2013
Route Intravenous Intravenous infusion of xenin-25 (4 pmoles x kg-1 x min-1) in 1% human albumin in normal saline” NCT00798915
Target NTSR1 “Xenin-25 (Xen) is a 25-amino acid neurotensin-related peptide that activates neurotensin receptor-1 (NTSR1).” PMID 24183983 Oct 2013