Drugs / Golvatinib
last change Sep 2017 re-read 2 minutes ago

Golvatinib

Small molecule targets KDR, MET via inhibition

Developed for
cancer · gastric cancer · head and neck squamous cell carcinoma
Investigated by
Eisai Inc. · Quintiles, Inc.

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT01428141 Sep 2011 → Jan 2013 gastric cancer Eisai Inc. Completed No outcome recorded
Phase 1 NCT02533102 Nov → Dec 2010 Eisai Inc. Completed No outcome recorded
Phase 1 NCT00921869 Oct 2009 → Jun 2011 cancer Eisai Inc. Completed No outcome recorded
Phase 1 NCT00869895 Mar 2009 → Aug 2012 cancer Eisai Inc. Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT01355302 Nov 2011 → Apr 2013 Eisai Inc. Terminated No outcome recorded
Phase 1/2 NCT01433991 Oct 2011 → Mar 2015 cancer Eisai Inc. Terminated No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/2 NCT01332266 Comparator Sep 2011 → Jan 2016 head and neck squamous cell carcinoma Eisai Inc. Completed No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as Golvatinib ClinicalTrials.gov intervention name — accepted as the source's own label NCT01433991
Known as E-7050 (GOLVATINIB) ChEMBL registry synonym — accepted as the source's own label CHEMBL3039525
Known as E7050 “This study is designed to first evaluate the effect of food on E7050's pharmacokinetic parameters following the administration of single 100 mg oral doses of E7050 tablet to...” NCT02533102
5

NCT00921869

NCT01428141

NCT00869895

NCT01332266

NCT01355302

Known as ER-396901-08 ChEMBL registry synonym — accepted as the source's own label CHEMBL3039525
Known as GOLVATINIB (E7050) ChEMBL registry synonym — accepted as the source's own label CHEMBL3039525
Known as GOLVATINIB TARTRATE ChEMBL registry synonym — accepted as the source's own label CHEMBL3039525
Action Inhibit “Vascular endothelial growth factor receptor 2 inhibitor” CHEMBL3039525
1

“Hepatocyte growth factor receptor inhibitor” CHEMBL3039525

Modality Small molecule CHEMBL3039525
Route Oral “given orally” NCT00869895
Target KDR “Vascular endothelial growth factor receptor 2 inhibitor” CHEMBL3039525
Target MET “Hepatocyte growth factor receptor inhibitor” CHEMBL3039525