Drugs / Afimetoran
last change Jun 2026 re-read 2 minutes ago

Afimetoran

also known as BMS-986256

Small molecule targets TLR7, TLR8 via inhibition

Developed for
cutaneous lupus erythematosus · systemic lupus erythematosus
Investigated by
Bristol-Myers Squibb

Trials 11 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 110 trials
Phase 1 NCT05866627 Jul → Sep 2023 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT05901714 Jun 2023 → Apr 2024 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT04941755 Jun → Sep 2021 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT04493541 Aug 2020 → Apr 2023 cutaneous lupus erythematosus Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT04470778 Jul 2020 → Mar 2021 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT04269356 Feb 2020 → Mar 2021 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT04016753 Aug 2019 → Feb 2020 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT04039373 Jul → Sep 2019 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT03950960 May → Jul 2019 Bristol-Myers Squibb Completed No outcome recorded
Phase 1 NCT03634995 Aug 2018 → Oct 2019 Bristol-Myers Squibb Completed No outcome recorded
Phase 21 trial
Phase 2 NCT04895696 Oct 2021 → Jun 2026 overdue systemic lupus erythematosus Bristol-Myers Squibb Active not recruiting No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as Afimetoran ClinicalTrials.gov intervention name — accepted as the source's own label NCT04895696
2

NCT05866627

NCT05901714

Known as BMS-986256 “An Open-label, Single-sequence, Drug-drug Interaction Study in Healthy Participants to Assess the Effect of Phenytoin on the Pharmacokinetics of a Single Oral Dose of...” NCT05901714
8

NCT04941755

NCT03950960

NCT04016753

NCT04039373

NCT04470778

NCT04493541

NCT04269356

NCT03634995

Action Inhibit “Toll-like receptor 8 inhibitor” CHEMBL4650329
1

“Toll-like receptor 7 inhibitor” CHEMBL4650329

Modality Small molecule CHEMBL4650329
Target TLR7 “Toll-like receptor 7 inhibitor” CHEMBL4650329
Target TLR8 “Toll-like receptor 8 inhibitor” CHEMBL4650329