Drugs / Latanoprostene bunod
last change Aug 2023 re-read 2 minutes ago

Latanoprostene bunod

Small molecule targets PTGFR via activation

Developed for
ocular hypertension · open-angle glaucoma · glaucoma
Investigated by
Bausch & Lomb Incorporated · University of California, San Diego

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved US (FDA) VYZULTA 2017-11-02 fda.gov

Trials 8 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT01895985 Jul → Aug 2013 Bausch & Lomb Incorporated Completed No outcome recorded
Phase 22 trials
Phase 2 NCT01707381 Nov 2012 → Dec 2013 ocular hypertension, open-angle glaucoma Bausch & Lomb Incorporated Completed No outcome recorded
Phase 2 NCT01223378 Dec 2010 → Dec 2011 Bausch & Lomb Incorporated Completed No outcome recorded
Phase 33 trials
Phase 3 NCT01895972 Jul 2013 → Apr 2015 glaucoma, ocular hypertension Bausch & Lomb Incorporated Completed No outcome recorded
Phase 3 NCT01749904 Jan 2013 → Jun 2015 ocular hypertension, open-angle glaucoma Bausch & Lomb Incorporated Completed No outcome recorded
Phase 3 NCT01749930 Jan 2013 → May 2015 ocular hypertension, open-angle glaucoma Bausch & Lomb Incorporated Completed No outcome recorded
Phase 41 trial
Phase 4 NCT04140279 May 2022 → Aug 2023 ocular hypertension Bausch & Lomb Incorporated Withdrawn No outcome recorded
Phase not applicable1 trial
NCT03931317 Dec 2018 → May 2021 ocular hypertension, open-angle glaucoma University of California, San Diego Completed No outcome recorded

Evidence & citations 12 cited values

Every value below carries the sentence it was read from. 11 sources stand behind the page.

FieldValueCited text
Known as Latanoprostene bunod “Comparison of Latanoprostene Bunod 0.024% and Timolol Maleate 0.5% in Open-Angle Glaucoma or Ocular Hypertension: The LUNAR Study.” PMID 27210275 May 2016
4

NCT01895985

NCT03931317

NCT04140279

NCT01895972

Known as BOL-303259-X ClinicalTrials.gov intervention name — accepted as the source's own label NCT01749904
2

NCT01707381

NCT01223378

Known as Latanoprosteno bunod ChEMBL registry synonym — accepted as the source's own label CHEMBL2364612
Known as LBN “PURPOSE: To compare the intraocular pressure (IOP)-lowering effect of latanoprostene bunod (LBN) 0.024% with timolol maleate 0.5% in subjects with open-angle glaucoma (OAG) or...” PMID 27210275 May 2016
Known as NCX 116 ChEMBL registry synonym — accepted as the source's own label CHEMBL2364612
Known as PF-3187207 ChEMBL registry synonym — accepted as the source's own label CHEMBL2364612
Known as Vesneo ChEMBL registry synonym — accepted as the source's own label CHEMBL2364612
Known as Vyzulta ChEMBL registry synonym — accepted as the source's own label CHEMBL2364612
Action Activate “prostaglandin F2α receptor agonist” PMID 26563323 Nov 2015
1

“Prostanoid FP receptor agonist” CHEMBL2364612

Modality Small molecule CHEMBL2364612
Route Topical “Subjects instilled one drop of study medication in the study eye” PMID 25488946 Dec 2014
Target PTGFR “Prostanoid FP receptor agonist” CHEMBL2364612