Drugs / MK-0736
last change Mar 2011 re-read 2 minutes ago

MK-0736

Small molecule targets HSD11B1 via inhibition

Developed for
hypertensive disorder · type 2 diabetes mellitus · peripheral vascular disease
Investigated by
Merck Sharp & Dohme LLC

Trials 2 · a red edge is where a trial was stopped

2006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT00806585 Dec 2008 → Mar 2010 hypertensive disorder, type 2 diabetes mellitus Merck Sharp & Dohme LLC Terminated No outcome recorded
Phase 2 NCT00274716 Nov 2005 → Jan 2007 hypertensive disorder Merck Sharp & Dohme LLC Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT00679055 Comparator Mar 2007 → Aug 2008 peripheral vascular disease Merck Sharp & Dohme LLC Terminated No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 5 sources stand behind the page.

FieldValueCited text
Known as MK0736 “This study evaluated the antihypertensive efficacy and safety of two 11β-HSD1 inhibitors, MK-0736 and MK-0916, in overweight-to-obese hypertensive patients.” PMID 21419745 Mar 2011
4

“Dose-ranging Study to Evaluate the Effectiveness and Tolerability of MK0736 in Patients With Type 2 Diabetes Mellitus (T2DM) and Hypertension (0736-007)” NCT00806585

NCT00274716

NCT00679055

NCT00806585

Action Inhibit “two 11β-HSD1 inhibitors” PMID 21419745 Mar 2011
Modality Small molecule CHEMBL1761322
Route Oral “Participants will be orally administered 7 mg of MK-0736 once daily for 12 weeks” NCT00679055
Target HSD11B1 “This study evaluated the antihypertensive efficacy and safety of two 11β-HSD1 inhibitors, MK-0736 and MK-0916, in overweight-to-obese hypertensive patients.” PMID 21419745 Mar 2011