Drugs / AB-106
last change Apr 2026 re-read 2 minutes ago

AB-106

also known as Taletrectinib · DS-6051b

Small molecule targets ALK, DDR1, LTK, ROS1 via inhibition

Developed for
non-small cell lung carcinoma · breast cancer · bronchogenic carcinoma · neoplasm
Investigated by
Nuvation Bio Inc. · AnHeart Therapeutics Inc. · Megan Kruse, MD

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT05609929 Nov 2022 → Jan 2023 Nuvation Bio Inc. Completed No outcome recorded
Phase 1 NCT05357820 Jul → Dec 2021 cancer Nuvation Bio Inc. Completed No outcome recorded
Phase 1 NCT05357911 Jul → Aug 2021 cancer Nuvation Bio Inc. Completed No outcome recorded
Phase 24 trials
Phase 2 NCT06214793 Oct 2026 → Jan 2030 breast cancer Megan Kruse, MD Suspended No outcome recorded
Phase 2 NCT04919811 Sep 2021 → Jun 2025 overdue non-small cell lung carcinoma Nuvation Bio Inc. Active not recruiting No outcome recorded
Phase 2 NCT04617054 Jun 2021 → Dec 2024 neoplasm Nuvation Bio Inc. Terminated No outcome recorded
Phase 2 NCT04395677 Jul 2020 → Jun 2024 overdue non-small cell lung carcinoma Nuvation Bio Inc. Active not recruiting No outcome recorded
Phase 31 trial
Phase 3 NCT06564324 Nov 2024 → Jan 2029 expected non-small cell lung carcinoma Nuvation Bio Inc. Recruiting No outcome recorded
Phase not stated1 trial
NCT06841874 bronchogenic carcinoma, non-small cell lung carcinoma Nuvation Bio Inc. No longer available No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 3 NCT07154706 Comparator Aug 2025 → Aug 2030 expected non-small cell lung carcinoma Nuvation Bio Inc. Recruiting No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as AB-106 “Former Name(s) or Alias(es): AB-106.” NCT07154706
5

NCT05357820

NCT04617054

NCT05357911

NCT05609929

NCT04395677

Known as DS-6051b “Taletrectinib (AB-106/DS-6051b) is a potent, highly selective, orally bioavailable ROS1 and TRK family inhibitor” NCT06214793
Known as Taletrectinib ClinicalTrials.gov intervention name — accepted as the source's own label NCT04919811
4

NCT07154706

NCT06841874

NCT06564324

NCT06214793

Action Inhibit “ROS1 tyrosine kinase inhibitor (TKI)” PMID 42013573 Apr 2026
Modality Small molecule “ROS1 tyrosine kinase inhibitor (TKI)” PMID 42013573 Apr 2026
Route Oral “once-daily oral taletrectinib 600 mg” PMID 40179330 Apr 2025
Target ROS1 ROS1 tyrosine kinase inhibitor (TKI)” PMID 42013573 Apr 2026