Drugs / dexmecamylamine

Trials 19 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 19 trials
Phase 1 NCT01500018 Jan → Apr 2012 substance abuse AstraZeneca Withdrawn No outcome recorded
Phase 1 NCT01458899 Nov 2011 → Jan 2012 AstraZeneca Completed No outcome recorded
Phase 1 NCT01403922 Aug 2011 → Aug 2012 hypertensive disorder AstraZeneca Terminated No outcome recorded
Phase 1 NCT01392820 Jul → Oct 2011 AstraZeneca Completed No outcome recorded
Phase 1 NCT01359618 Jun 2011 → Apr 2012 AstraZeneca Terminated No outcome recorded
Phase 1 NCT01239771 Jan → May 2011 AstraZeneca Completed No outcome recorded
Phase 1 NCT01240967 Nov 2010 → Jul 2011 impaired renal function disease AstraZeneca Completed No outcome recorded
Phase 1 NCT01175564 Jul → Sep 2010 AstraZeneca Completed No outcome recorded
Phase 1 NCT01145768 Jun → Aug 2010 AstraZeneca Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00899977 May → Aug 2009 resistant hypertension Targacept Inc. Terminated No outcome recorded
Phase 24 trials
Phase 2 NCT04263623 Jan → Dec 2020 hyperhidrosis palmaris ET plantaris, isolated hyperchlorhidrosis Atacama Therapeutics Unknown No outcome recorded
Phase 2 NCT03404570 Dec 2017 → Jan 2019 hyperhidrosis palmaris ET plantaris Atacama Therapeutics Completed No outcome recorded
Phase 2 NCT01868516 May 2013 → Jun 2014 overactive bladder Targacept Inc. Completed No outcome recorded
Phase 2 NCT01288079 Feb 2011 → Aug 2012 major depressive disorder AstraZeneca Terminated No outcome recorded
Phase 35 trials
Phase 3 NCT01180400 Sep 2010 → Sep 2011 major depressive disorder AstraZeneca Completed No outcome recorded
Phase 3 NCT01197508 Sep 2010 → Jan 2012 major depressive disorder AstraZeneca Completed No outcome recorded
Phase 3 NCT01152554 Jun 2010 → Feb 2012 major depressive disorder AstraZeneca Completed No outcome recorded
Phase 3 NCT01157078 Jun 2010 → Nov 2011 major depressive disorder AstraZeneca Completed No outcome recorded
Phase 3 NCT01153347 Jun 2010 → Jan 2012 major depressive disorder AstraZeneca Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT00692445 Comparator Jun 2008 → May 2009 major depressive disorder Targacept Inc. Completed No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 25 sources stand behind the page.

FieldValueCited text
Known as dexmecamylamine “This paper reports the efficacy and tolerability of the nicotinic channel modulator TC-5214 (dexmecamylamine) as adjunct therapy for patients with major depressive disorder who...” PMID 24507016 Dec 2013
6

“Two Phase III randomised double-blind studies of fixed-dose TC-5214 (dexmecamylamine) adjunct to ongoing antidepressant therapy in patients with major depressive disorder and...” PMID 25602163 Jan 2015

“TC-5214 (dexmecamylamine) is a nicotinic channel modulator that has previously been evaluated for treatment of major depression disorder (MDD) and is currently being evaluated...” PMID 24408516 Jan 2014

“nicotinic channel modulator dexmecamylamine (TC-5214)” PMID 25514064 Feb 2015

NCT01868516

NCT04263623

NCT03404570

Known as Dexmecamilamina ChEMBL registry synonym — accepted as the source's own label CHEMBL2103881
Known as Dexmecamylamine HCl “Oral tablet containing 2 mg of active drug, dexmecamylamine HCl.” NCT04263623
1

“Oral tablet containing 2 mg of active drug, dexmecamylamine HCl.” NCT03404570

Known as DEXMECAMYLAMINE HYDROCHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL2103881
Known as Mecamylamine s-(+)-form hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL2103881
Known as NIH-11008 ChEMBL registry synonym — accepted as the source's own label CHEMBL2103881
Known as S-Mecamylamine “A Phase IIb, Randomized, Double-Blind, Placebo-Controlled, Active Controlled, Parallel Group, Multicenter Study to Assess the Safety and Efficacy of 2 Fixed Dose Groups of...” NCT01288079
7

“A Multicenter, Randomized, Double-Blind Parallel Group Placebo-Controlled Phase III, Efficacy and Safety Study of 3 Fixed Dose Groups of TC-5214 (S-mecamylamine) as an Adjunct...” NCT01197508

“A Multicenter, Randomized, Double-Blind, Parallel Group, Placebo-Controlled, Phase III Efficacy and Safety Study of TC-5214 (S-mecamylamine) in Flexible Doses as an Adjunct to...” NCT01180400

“An Open-Label, Multi-Center, Phase I Study To Compare the Pharmacokinetics of a Single Oral Dose of TC-5214 (S-Mecamylamine) in Subjects With Renal Impairment With Subjects...” NCT01240967

“after a single and repeated oral doses of TC-5214 (S-mecamylamine) in healthy male Japanese subjects” NCT01175564

“Oral TC-5214 (S-Mecamylamine) After Administration of Single and Multiple Ascending Doses” NCT01145768

“TC-5214 (S-mecamylamine) as an Adjunct to an Antidepressant” NCT01152554

“TC-5214 (S-Mecamylamine)” NCT01458899

Known as TC-5214 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00692445
16

NCT01359618

NCT01239771

NCT01175564

NCT01392820

NCT01153347

NCT01403922

NCT01157078

NCT01240967

NCT01145768

NCT00899977

NCT01152554

NCT01458899

NCT01197508

NCT01180400

NCT01500018

NCT01288079

Known as TC-5214-23 “TC-5214 (as TC-5214-23) will be provided as white, opaque, hard-gelatin capsules in strengths of 1, 2, and 4 mg.” NCT00692445
Modality Other / unclassified “nicotinic channel modulator dexmecamylamine (TC-5214)” PMID 25514064 Feb 2015
Route Oral “Concentration-time profiles of TC-5214 after either single or multiple oral doses of TC-5214 was described by a one-compartment model with first-order absorption with lag time...” PMID 24408516 Jan 2014