Drugs / Pamiparib
last change Aug 2026 re-read 2 minutes ago

Pamiparib

also known as BGB-290

Small molecule targets PARP1, PARP2 via inhibition

Developed for
ovarian cancer · cancer · castration-resistant prostate carcinoma · glioblastoma · grade II glioma · grade III glioma · adult glioblastoma · brain cancer
+18 more · carcinosarcoma · clear cell papillary renal cell carcinoma · collecting duct carcinoma · gastric cancer · head and neck squamous cell carcinoma · Her2-receptor negative breast cancer · hereditary leiomyomatosis and renal cell cancer · hereditary papillary renal cell carcinoma · malignant epithelial tumor of ovary · metastatic prostate carcinoma · non-small cell lung carcinoma · pharynx cancer · prostate cancer · refractory malignant neoplasm · salivary gland carcinoma · small cell lung carcinoma · triple-negative breast carcinoma · tubulocystic renal cell carcinoma
Investigated by
BeiGene · Sun Yat-sen University · BeiGene · Affiliated Hospital of Jiangnan University · Anhui Provincial Hospital · Australia New Zealand Gynaecological Oncology Group
+38 more · Bai-Rong Xia · Barrow Neurological Institute · BeOne Medicines · Chongqing University Cancer Hospital · Driven To Cure · European Organisation for Research and Treatment of Cancer - EORTC · First Affiliated Hospital Xi'an Jiaotong University · First Affiliated Hospital of Zhejiang University · Fudan University · Fujian Cancer Hospital · Hongqian Guo · Hubei Cancer Hospital · Hutchmed · Ivy Brain Tumor Center · Jonsson Comprehensive Cancer Center · M.D. Anderson Cancer Center · Myriad Genetic Laboratories, Inc. · Myriad Genetics, Inc. · Nader Sanai · Nanjing First Hospital, Nanjing Medical University · National Cancer Institute (NCI) · Peking Union Medical College · Peking University Cancer Hospital & Institute · Peking University Hospital of Stomatology · Peking University Shenzhen Hospital · Peter MacCallum Cancer Centre, Australia · Qilu Hospital of Shandong University · Shandong Cancer Hospital and Institute · Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins · Sun Yat-sen University Cancer Center · The Affiliated Nanjing Drum Tower Hospital of Nanjing University Medical School · The First Affiliated Hospital of Soochow University · The First Affiliated Hospital of Xiamen University · Tongji Hospital · Union Hospital, Tongji Medical College · University of California, San Francisco · University of Chicago · Zhejiang Cancer Hospital

Trials 34 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT04614909 Jan 2021 → Jul 2023 adult glioblastoma Nader Sanai Completed No outcome recorded
Phase 19 trials
Phase 1 NCT05526924 Mar 2023 → Jan 2028 expected head and neck squamous cell carcinoma, pharynx cancer University of Chicago Recruiting No outcome recorded
Phase 1 NCT05573373 Dec 2022 → Nov 2024 non-small cell lung carcinoma Affiliated Hospital of Jiangnan University Unknown No outcome recorded
Phase 1 NCT05038839 Feb 2022 → May 2026 refractory malignant neoplasm M.D. Anderson Cancer Center Completed No outcome recorded
Phase 1 NCT03991494 May → Oct 2019 cancer BeiGene Completed No outcome recorded
Phase 1 NCT03994211 May → Oct 2019 cancer BeiGene Completed No outcome recorded
Phase 1 NCT03749187 Apr 2019 → Jun 2026 overdue glioblastoma, grade II glioma, grade III glioma University of California, San Francisco Active not recruiting No outcome recorded
Phase 1 NCT03150810 Jun 2017 → May 2023 BeiGene Completed No outcome recorded
Phase 1 NCT02660034 Feb 2016 → Sep 2020 cancer BeiGene Completed No outcome recorded
Phase 1 NCT02361723 Jul 2014 → Sep 2019 BeiGene Completed No outcome recorded
Phase 1/24 trials
Phase 1/2 NCT05494580 Sep 2022 → Jun 2024 fallopian tube carcinosarcoma, ovarian carcinoma, primary peritoneal carcinoma Sun Yat-sen University Completed No outcome recorded
Phase 1/2 NCT03914742 Feb 2020 → Oct 2023 glioblastoma, grade II glioma, grade III glioma Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins Completed No outcome recorded
Phase 1/2 NCT03150862 Jul 2017 → Mar 2021 brain cancer BeiGene Completed No outcome recorded
Phase 1/2 NCT03333915 Dec 2016 → Aug 2020 ovarian cancer, triple-negative breast carcinoma BeiGene Completed No outcome recorded
Phase 218 trials
Phase 2 NCT06692491 Jan 2025 → Dec 2027 expected Peking University Shenzhen Hospital Not yet recruiting No outcome recorded
Phase 2 NCT06387056 Apr 2024 → Apr 2026 overdue metastatic prostate carcinoma The First Affiliated Hospital of Xiamen University Recruiting No outcome recorded
Phase 2 NCT06145308 Aug 2023 → Jul 2028 expected salivary gland carcinoma Peking Union Medical College Recruiting No outcome recorded
Phase 2 NCT05669768 Jan 2023 → Jul 2024 ovarian cancer Sun Yat-sen University Unknown No outcome recorded
Phase 2 NCT05652283 Nov 2022 → May 2024 overdue ovarian cancer Bai-Rong Xia Active not recruiting No outcome recorded
Phase 2 NCT05489926 Aug 2022 → Jun 2024 malignant epithelial tumor of ovary Zhejiang Cancer Hospital Unknown No outcome recorded
Phase 2 NCT05044871 Jul 2022 → Feb 2025 ovarian cancer Tongji Hospital Completed No outcome recorded
Phase 2 NCT05483543 Jun 2022 → Dec 2024 small cell lung carcinoma Fudan University Unknown No outcome recorded
Phase 2 NCT05327621 May 2022 → Mar 2025 castration-resistant prostate carcinoma Sun Yat-sen University Unknown No outcome recorded
Phase 2 NCT04796454 May 2022 → Jul 2026 European Organisation for Research and Treatment of Cancer - EORTC Withdrawn No outcome recorded
Phase 32 trials
Phase 3 NCT04164199 Dec 2019 → May 2026 cancer BeOne Medicines Completed No outcome recorded
Phase 3 NCT03519230 May 2018 → Dec 2025 overdue ovarian cancer BeiGene Active not recruiting No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 36 sources stand behind the page.

FieldValueCited text
Known as Pamiparib Pamiparib (BGB-290) Was Used in EGFR-TkIs Resistant Non-small Cell Lung Cancer” NCT05573373
30

“Available drugs include olaparib, fluzoparib, pamiparib, talazoparib ect.” NCT05406999

“60mg pamiparib (BGB-290) PO BID” NCT03749187

pamiparib 60 mg PO bid” NCT06145308

NCT03150862

NCT03427814

NCT04796454

NCT05489926

NCT02660034

NCT05652283

NCT05494580

NCT03994211

NCT05669768

NCT05526924

NCT05483543

NCT05038839

NCT03991494

NCT06387056

NCT03333915

NCT04603365

NCT05044871

NCT06692491

NCT03519230

NCT05376722

NCT04164199

NCT03712930

NCT04985721

NCT03150810

NCT04614909

NCT05327621

NCT03933761

Known as BGB-290 “A Phase 1, Open-label, Parallel-group, Fixed-sequence Study to Investigate the Effect of the CYP3A Inducer Rifampin and the CYP3A Inhibitor Itraconazole on the Pharmacokinetics...” NCT03994211
5

“Pamiparib (BGB-290)” NCT03933761

NCT03914742

NCT03749187

NCT03575065

NCT02361723

Action Inhibit “pamiparib, an oral PARP 1/2 inhibitor” PMID 31378459 Aug 2019
Modality Small molecule “Pamiparib is a small molecule inhibitor selectivity for both PARP1 and PARP2.” NCT05494580
Route Oral “20, 40, or 60 mg oral pamiparib twice daily” PMID 31378459 Aug 2019
Target PARP1 “excellent selectivity for both PARP1 and PARP2” PMID 32652442 Jul 2020
Target PARP2 “excellent selectivity for both PARP1 and PARP2PMID 32652442 Jul 2020