Drugs / Zeprumetostat

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT07692529 Aug 2026 → Dec 2027 expected Institute of Hematology & Blood Diseases Hospital, China Not yet recruiting No outcome recorded
Phase 1/25 trials
Phase 1/2 NCT07706959 Jul 2026 → Jan 2028 expected peripheral T-cell lymphoma, not otherwise specified Ruijin Hospital Not yet recruiting No outcome recorded
Phase 1/2 NCT07643805 Jun 2026 → Jan 2028 expected diffuse large B-cell lymphoma The First Affiliated Hospital with Nanjing Medical University Not yet recruiting No outcome recorded
Phase 1/2 NCT07502768 Apr 2026 → Dec 2027 expected extranodal nasal NK/T cell lymphoma, mature T-cell and NK-cell non-Hodgkin lymphoma Rong Tao Recruiting No outcome recorded
Phase 1/2 NCT07493330 Mar 2026 → Dec 2029 expected refractory malignant neoplasm Ruijin Hospital Not yet recruiting No outcome recorded
Phase 1/2 NCT07339527 Jan 2026 → Jan 2028 expected mature T-cell and NK-cell non-Hodgkin lymphoma Sun Yat-sen University Not yet recruiting No outcome recorded
Phase 23 trials
Phase 2 NCT07555470 Apr 2026 → Dec 2029 expected follicular lymphoma Institute of Hematology & Blood Diseases Hospital, China Recruiting No outcome recorded
Phase 2 NCT07372352 Jan 2026 → Jan 2028 expected peripheral T-cell lymphoma, not otherwise specified The First Affiliated Hospital of Soochow University Recruiting No outcome recorded
Phase 2 NCT07339553 Jan 2026 → Jan 2029 expected ovarian carcinoma Peking University Third Hospital Not yet recruiting No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 10 sources stand behind the page.

FieldValueCited text
Known as Zeprumetostat “Phase 2: Zeprumetostat Tablets in Combination with Fuzuloparib Dose: Zeprumetostat Tablets 250 mg, bid, po, Fuzuloparib 100 mg, bid, po.” NCT07339553
8

“Single-Arm Clinical Study of Zeprumetostat in Combination with Glofitamab + GemOx in Patients with Relapsed/ Refractory DLBCL” NCT07643805

NCT07493330

NCT07502768

NCT07555470

NCT07339527

NCT07692529

NCT07706959

NCT07372352

Known as SHR2554 “Zeprumetostat (SHR2554), an oral EZH2 inhibitor, administered twice daily.” NCT07502768
Action Inhibit “EZH2 inhibitor Zeprumetostat” NCT07339527
Modality Small molecule CHEMBL5939817
Route Oral “350mg, po, bid” NCT07339527
Target EZH2 EZH2 inhibitor Zeprumetostat” NCT07339527