Drugs / Fenebrutinib
last change Jan 2026 re-read 2 minutes ago

Fenebrutinib

also known as GDC-0853 · G-02599853 · RG-7845 · RO-7010939

Small molecule targets BTK via inhibition

Developed for
multiple sclerosis · rheumatoid arthritis · systemic lupus erythematosus · chronic urticaria · diffuse large B-cell lymphoma · primary progressive multiple sclerosis · urticaria
Investigated by
Genentech, Inc. · Hoffmann-La Roche

Trials 17 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT03596632 Jul → Aug 2018 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT03290703 Apr 2017 → Oct 2018 Genentech, Inc. Completed No outcome recorded
Phase 1 NCT03174041 Apr → Jun 2017 Genentech, Inc. Completed No outcome recorded
Phase 1 NCT03188783 Jan → Aug 2017 Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT02699710 Sep 2015 → May 2016 Genentech, Inc. Completed No outcome recorded
Phase 1 NCT01991184 Dec 2013 → Mar 2022 diffuse large B-cell lymphoma Genentech, Inc. Completed No outcome recorded
Phase 28 trials
Phase 2 NCT07161258 Oct 2025 → Jun 2027 expected multiple sclerosis Hoffmann-La Roche Recruiting No outcome recorded
Phase 2 NCT05119569 Mar 2022 → Mar 2023 overdue multiple sclerosis Hoffmann-La Roche Active not recruiting No outcome recorded
Phase 2 NCT03693625 Sep 2018 → Oct 2019 urticaria Genentech, Inc. Terminated No outcome recorded
Phase 2 NCT03407482 Jan 2018 → Nov 2019 systemic lupus erythematosus Genentech, Inc. Terminated No outcome recorded
Phase 2 NCT03137069 May 2017 → Sep 2019 chronic urticaria Genentech, Inc. Completed No outcome recorded
Phase 2 NCT02908100 Jan 2017 → May 2019 systemic lupus erythematosus Genentech, Inc. Completed No outcome recorded
Phase 2 NCT02983227 Nov 2016 → Jul 2019 rheumatoid arthritis Genentech, Inc. Completed No outcome recorded
Phase 2 NCT02833350 Sep 2016 → Jul 2018 rheumatoid arthritis Genentech, Inc. Completed No outcome recorded
Phase 33 trials
Phase 3 NCT04586023 Mar 2021 → Sep 2025 overdue multiple sclerosis Hoffmann-La Roche Active not recruiting No outcome recorded
Phase 3 NCT04586010 Mar 2021 → Jan 2026 overdue multiple sclerosis Hoffmann-La Roche Active not recruiting No outcome recorded
Phase 3 NCT04544449 Oct 2020 → Sep 2025 overdue primary progressive multiple sclerosis Hoffmann-La Roche Active not recruiting No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 19 sources stand behind the page.

FieldValueCited text
Known as Fenebrutinib Fenebrutinib (GDC-0853) is a noncovalent, oral, and highly selective inhibitor of Bruton's tyrosine kinase (BTK).” PMID 34042314 Aug 2021
6

NCT04586023

NCT04586010

NCT03596632

NCT07161258

NCT05119569

NCT04544449

Known as G-02599853 ChEMBL registry synonym — accepted as the source's own label CHEMBL4065122
Known as GDC-0853 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02699710
10

NCT03137069

NCT02983227

NCT03407482

NCT03188783

NCT02833350

NCT02908100

NCT03693625

NCT03174041

NCT01991184

NCT03290703

Known as RG-7845 ChEMBL registry synonym — accepted as the source's own label CHEMBL4065122
Known as RO-7010939 ChEMBL registry synonym — accepted as the source's own label CHEMBL4065122
Action Inhibit inhibitor of Bruton's tyrosine kinase (BTK)” PMID 34042314 Aug 2021
Modality Small molecule CHEMBL4065122
Route Oral “administered orally” NCT02699710
Target BTK “inhibitor of Bruton's tyrosine kinase (BTK)” PMID 34042314 Aug 2021