Drugs / Xevinapant

Trials 18 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 110 trials
Phase 1 NCT06463184 Jul 2024 → Jun 2027 malignant glioma H. Lee Moffitt Cancer Center and Research Institute Withdrawn No outcome recorded
Phase 1 NCT06110195 Jan 2024 → May 2025 head and neck squamous cell carcinoma University of Chicago Terminated No outcome recorded
Phase 1 NCT06056310 Jan → Aug 2024 head and neck cancer EMD Serono Research & Development Institute, Inc. Terminated No outcome recorded
Phase 1 NCT05519540 Sep 2022 → Apr 2023 Merck Healthcare KGaA, Darmstadt, Germany, an affiliate of Merck KGaA, Darmstadt, Germany Completed No outcome recorded
Phase 1 NCT04962724 Aug → Nov 2021 Debiopharm International SA Completed No outcome recorded
Phase 1 NCT03871959 Sep 2019 → May 2022 colon adenocarcinoma, pancreatic adenocarcinoma, rectum adenocarcinoma Centre Leon Berard Completed No outcome recorded
Phase 1 NCT03270176 Oct 2017 → Mar 2022 non-small cell lung carcinoma Debiopharm International SA Completed No outcome recorded
Phase 1 NCT01930292 Apr 2013 → Mar 2016 cancer Debiopharm International SA Terminated No outcome recorded
Phase 1 NCT01265199 Feb 2011 → Jan 2013 acute myeloid leukemia Ascenta Therapeutics Terminated No outcome recorded
Phase 1 NCT01078649 Mar 2010 → Apr 2014 cancer, lymphoma Debiopharm International SA Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT04122625 Apr 2019 → Apr 2022 cancer Debiopharm International SA Completed No outcome recorded
Phase 23 trials
Phase 2 NCT06084845 Apr 2024 → May 2028 hypopharynx squamous cell carcinoma, laryngeal squamous cell carcinoma, oral cavity squamous cell carcinoma, oropharynx squamous cell carcinoma ECOG-ACRIN Cancer Research Group Withdrawn No outcome recorded
Phase 2 NCT06145412 Nov 2023 → Nov 2026 expected head and neck cancer Memorial Sloan Kettering Cancer Center Active not recruiting No outcome recorded
Phase 2 NCT05724602 Nov 2023 → Jul 2029 head and neck squamous cell carcinoma European Organisation for Research and Treatment of Cancer - EORTC Suspended No outcome recorded
Phase 33 trials
Phase 3 NCT05930938 Dec 2023 → Sep 2024 head and neck squamous cell carcinoma Groupe Oncologie Radiotherapie Tete et Cou Terminated No outcome recorded
Phase 3 NCT05386550 Oct 2022 → Aug 2024 head and neck squamous cell carcinoma EMD Serono Research & Development Institute, Inc. Terminated No outcome recorded
Phase 3 NCT04459715 Aug 2020 → Sep 2024 head and neck squamous cell carcinoma EMD Serono Research & Development Institute, Inc. Terminated No outcome recorded
Phase not applicable1 trial
NCT02022098 Oct 2013 → Jul 2020 head and neck squamous cell carcinoma Debiopharm International SA Completed No outcome recorded

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 20 sources stand behind the page.

FieldValueCited text
Known as Xevinapant “A Study of Xevinapant With Cisplatin and Radiation Therapy After Surgery in People With Head and Neck Cancer” NCT06145412
10

NCT06463184

NCT04962724

NCT06110195

NCT06084845

NCT06056310

NCT05930938

NCT04459715

NCT05519540

NCT05724602

NCT05386550

Known as AT-406 “compound Debio 1143 (AT-406), a small molecule second mitochondria-derived activator of caspase C (Smac) mimetic” NCT01078649
1

NCT01265199

Known as D-1143 ChEMBL registry synonym — accepted as the source's own label CHEMBL2158051
Known as DEBIO1143 “Debio 1143 is an investigational, oral monovalent second mitochondrial-derived activator of caspases (SMAC) mimetic designed to promote programmed cell death (apoptosis) in...” NCT03871959
10

“PURPOSE: To assess safety/tolerability, pharmacokinetics (PK), pharmacodynamics (PD), and antitumor activity of DEBIO1143, an antagonist of inhibitor apoptosis proteins.” PMID 25716544 Feb 2015

“Adaptive doses of Debio1143 oral capsules, between 50 and 400 mg until the recommended dose (RD) is determined.” NCT01930292

“Xevinapant (Debio 1143) administrated as oral solution from Day 1 to 14, every 21-day cycle.” NCT04459715

“Xevinapant (Debio 1143)” NCT05519540

“Drug: DEBIO1143NCT03871959

NCT02022098

NCT01930292

NCT03270176

NCT01078649

NCT04122625

Known as IAP INHIBITOR AT-406 ChEMBL registry synonym — accepted as the source's own label CHEMBL2158051
Known as MSC2735845A ChEMBL registry synonym — accepted as the source's own label CHEMBL2158051
Known as SM-406 ChEMBL registry synonym — accepted as the source's own label CHEMBL2158051
Action Inhibit inhibiting XIAP (X linked IAP)” NCT01078649
Modality Small molecule “a small molecule second mitochondria-derived activator of caspase C (Smac) mimetic” NCT01078649
Route Oral “when administered orally” NCT01078649
Target XIAP “inhibiting XIAP (X linked IAP)” NCT01078649