Drugs / Evacetrapib
last change May 2017 re-read 2 minutes ago

Evacetrapib

also known as LY2484595

Small molecule targets CETP via inhibition

Developed for
hyperlipidemia · cardiovascular disorder · hyperlipoproteinemia
Investigated by
Eli Lilly and Company · The Cleveland Clinic

Trials 26 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 120 trials
Phase 1 NCT02497391 Jul → Nov 2015 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT02365558 Jan → Apr 2015 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT02271425 Oct → Nov 2014 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT02226653 Sep 2014 → Apr 2015 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT02156492 Jun → Dec 2014 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT02161731 Jun → Sep 2014 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT02168803 May 2014 → Dec 2015 hyperlipidemia Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01958489 Oct 2013 → Jan 2014 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01908582 Jul → Sep 2013 Eli Lilly and Company Completed No outcome recorded
Phase 1 NCT01903434 Jul → Nov 2013 Eli Lilly and Company Completed No outcome recorded
Phase 22 trials
Phase 2 NCT01375075 Jun 2011 → Mar 2012 hyperlipidemia Eli Lilly and Company Completed No outcome recorded
Phase 2 NCT01105975 Apr 2010 → Jun 2011 hyperlipidemia Eli Lilly and Company Completed No outcome recorded
Phase 34 trials
Phase 3 NCT02260648 Jan → Nov 2015 hyperlipidemia Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT02260635 Nov 2014 → Jul 2015 hyperlipoproteinemia Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT02227784 Oct 2014 → Dec 2015 hyperlipidemia Eli Lilly and Company Terminated No outcome recorded
Phase 3 NCT01687998 Oct 2012 → Mar 2016 cardiovascular disorder Eli Lilly and Company Terminated No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 28 sources stand behind the page.

FieldValueCited text
Known as Evacetrapib “LY2484595 (evacetrapib): 200 milligrams (mg) of LY2484595 administered orally, one time only” NCT01450098
21

NCT01897493

NCT01836185

NCT01908582

NCT02260635

NCT01903434

NCT02271425

NCT02156492

NCT02497391

NCT02161731

NCT01958489

NCT02168803

NCT01736254

NCT01687998

NCT02227784

NCT01810432

NCT02260648

NCT02226653

NCT01825876

NCT01825889

NCT02365558

NCT01746732

Known as LY2484595 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01375075
4

NCT01450098

NCT01448824

NCT01537887

NCT01105975

Action Inhibit “The cholesteryl ester transfer protein inhibitor evacetrapib” PMID 28514624 May 2017
1

“Cholesteryl ester transfer protein inhibitor” CHEMBL2017179

Modality Small molecule CHEMBL2017179
Route Oral “Administered orally” NCT01448824
Target CETP “Cholesteryl ester transfer protein inhibitor” CHEMBL2017179