Drugs / APG-1387
last change Oct 2025 re-read 2 minutes ago

APG-1387

also known as APG-1387 (SMAC MIMETIC) · SM-1387

Small molecule

Developed for
chronic hepatitis B virus infection · neoplasm · pancreatic adenocarcinoma
Investigated by
Ascentage Pharma Group Inc. · HealthQuest Pharma Inc.

Trials 5 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT03585322 Jul 2018 → Oct 2021 chronic hepatitis B virus infection Ascentage Pharma Group Inc. Completed No outcome recorded
Phase 1 NCT03386526 Nov 2017 → Oct 2022 neoplasm Ascentage Pharma Group Inc. Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT04643405 Mar 2021 → Jun 2024 pancreatic adenocarcinoma Ascentage Pharma Group Inc. Terminated No outcome recorded
Phase 1/2 NCT04284488 Apr 2020 → Nov 2024 neoplasm Ascentage Pharma Group Inc. Terminated No outcome recorded
Phase 21 trial
Phase 2 NCT04568265 Jun 2020 → Oct 2022 chronic hepatitis B virus infection Ascentage Pharma Group Inc. Unknown No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 7 sources stand behind the page.

FieldValueCited text
Known as APG-1387 ClinicalTrials.gov intervention name — accepted as the source's own label NCT04284488
4

NCT03386526

NCT04568265

NCT04643405

NCT03585322

Known as APG-1387 (SMAC MIMETIC) ChEMBL registry synonym — accepted as the source's own label CHEMBL4594459
Known as SM-1387 ChEMBL registry synonym — accepted as the source's own label CHEMBL4594459
Action Inhibit “APG-1387 is a novel second mitochondria-derived activator of caspase (Smac) mimetic IAP inhibitor.” PMID 38790057 May 2024
Modality Small molecule “APG-1387 is a potent, bivalent small-molecule Inhibitor of Apoptosis Protein (IAP) antagonist.” NCT03386526
Route Intravenous “30 minute IV infusion” NCT03386526