Drugs / Tedizolid Phosphate
last change Apr 2025 re-read 2 minutes ago

Tedizolid Phosphate

also known as MK-1986 · TR-701

Small molecule

Developed for
gram-positive bacterial infections
Investigated by
Merck Sharp & Dohme LLC · Merck & Co., Inc.

Regulatory milestones approvals, filings & regulatory actions · 5 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (3) US (FDA) SIVEXTRO 2019-03-06 – 2025-04-04 fda.gov
Approved EU (EMA) Sivextro 2015-03-23 europa.eu
Approved US (FDA) SIVEXTRO 2014-06-20 fda.gov

Trials 8 · a red edge is where a trial was stopped

20082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 17 trials
Phase 1 NCT06609161 Jul → Aug 2024 Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT06733688 Mar → Apr 2022 Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT03217565 Feb 2019 → Mar 2023 gram-positive bacterial infections Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT02750761 May 2016 → Dec 2018 gram-positive bacterial infections Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 1 NCT01442831 Sep 2010 Merck & Co., Inc. Completed No outcome recorded
Phase 1 NCT00876655 Feb → Mar 2009 Merck & Co., Inc. Completed No outcome recorded
Phase 1 NCT00666601 Apr → Aug 2008 Merck & Co., Inc. Completed No outcome recorded
Phase 31 trial
Phase 3 NCT03176134 Jan 2019 → Jul 2023 Merck Sharp & Dohme LLC Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 9 sources stand behind the page.

FieldValueCited text
Known as tedizolid phosphate “Study TR701-108 was a relative bioavailability study in 12 subjects administered 150-mg tedizolid equivalents as TPD or tedizolid phosphate.” PMID 23926058 Aug 2013
7

Tedizolid phosphate is a novel antibacterial prodrug with potent activity against Gram-positive pathogens.” PMID 24875463 May 2014

“tedizolid (TR-700), the active moiety of the antimicrobial prodrug tedizolid phosphate (TR-701)” PMID 22584101 May 2012

NCT06609161

NCT02750761

NCT06733688

NCT03176134

NCT03217565

Known as MK-1986 “A Phase 1, Single- and Multiple-Dose Safety and Pharmacokinetic Study of Oral and IV Tedizolid Phosphate (MK-1986) in Inpatients Under 2 Years Old” NCT03217565
1

“different oral formulations of tedizolid phosphate (MK-1986)” NCT06609161

Known as TR-701 “tedizolid (TR-700), the active moiety of the antimicrobial prodrug tedizolid phosphate (TR-701)” PMID 22584101 May 2012
Modality Small molecule “a novel oxazolidinone” PMID 22584101 May 2012
Route Oral “Each subject enrolled in the Main study will receive a single oral dose of 600mg TR-701” NCT00666601