Drugs / ARQ761
last change May 2022 re-read 2 minutes ago

ARQ761

also known as β-LAPACHONE

Small molecule

Developed for
cancer · lymphoma · malignant pancreatic neoplasm
Investigated by
University of Texas Southwestern Medical Center · ArQule, Inc.

Trials 3 · a red edge is where a trial was stopped

2012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT03575078 Jun 2018 → May 2019 lymphoma University of Texas Southwestern Medical Center Withdrawn No outcome recorded
Phase 1 NCT02514031 Mar 2016 → May 2018 malignant pancreatic neoplasm University of Texas Southwestern Medical Center Terminated No outcome recorded
Phase 1 NCT01502800 Dec 2011 → Feb 2017 cancer University of Texas Southwestern Medical Center Completed No outcome recorded

Evidence & citations 4 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as ARQ761 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03575078
2

NCT01502800

NCT02514031

Known as β-LAPACHONE “PHASE 1 DOSE ESCALATION TRIAL OF β-LAPACHONE (ARQ761) IN COMBINATION WITH PARP INHIBITOR, OLAPARIB, FOR REFRACTORY, ADVANCED SOLID TUMORS” NCT03575078
Modality Small molecule “ARQ 761 is a β-lapachone (β-lap) analogue that exploits the unique elevation of NQO1 found in solid tumours to cause tumour-specific cell death.” PMID 30318513 Oct 2018
Route Intravenous “ARQ 761 will be administered intravenously” NCT01502800