Drugs / REDAFAMDASTAT
last change Jul 2022 re-read 2 minutes ago

REDAFAMDASTAT

also known as PF-04457845 · CPD 23 · PF-4457845

Small molecule targets FAAH via inhibition

Developed for
osteoarthritis, knee · post-traumatic stress disorder · cannabis dependence · Tourette syndrome
Investigated by
Pfizer

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT01092845 Apr → Jun 2010 Pfizer Completed No outcome recorded
Phase 1 NCT01002625 Nov 2009 → Jan 2010 Pfizer Terminated No outcome recorded
Phase 1 NCT00918164 May → Jul 2009 Pfizer Completed No outcome recorded
Phase 1 NCT00836082 Feb → Jul 2009 chronic pain syndrome Pfizer Completed No outcome recorded
Phase 22 trials
Phase 2 NCT02216097 Oct 2014 → Mar 2015 post-traumatic stress disorder Pfizer Terminated No outcome recorded
Phase 2 NCT00981357 Nov 2009 → May 2010 osteoarthritis, knee Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 4 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT01665573 Comparator Jul 2012 → Oct 2015 Yale University Completed No outcome recorded
Phase 11 trial
Phase 1 NCT02134080 Comparator May 2014 → Mar 2017 Tourette syndrome Yale University Terminated No outcome recorded
Phase 22 trials
Phase 2 NCT03386487 Comparator Jan 2019 → Jul 2022 cannabis dependence Yale University Completed No outcome recorded
Phase 2 NCT01618656 Comparator Sep 2012 → Mar 2016 cannabis dependence Yale University Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 11 sources stand behind the page.

FieldValueCited text
Known as REDAFAMDASTAT ChEMBL registry synonym — accepted as the source's own label CHEMBL1651534
Known as CPD 23 ChEMBL registry synonym — accepted as the source's own label CHEMBL1651534
Known as PF-04457845 “The efficacy, safety and tolerability of the FAAH Inhibitor PF-0447845 in reducing cannabis use will be studied in a 4-site randomized, double-blind, placebo-controlled,...” NCT03386487
10

NCT01665573

NCT01618656

NCT00981357

NCT00836082

NCT00918164

NCT01092845

NCT03386487

NCT02216097

NCT02134080

NCT01002625

Known as PF-4457845 ChEMBL registry synonym — accepted as the source's own label CHEMBL1651534
Action Inhibit “FAAH inhibitor” NCT00836082
Modality Small molecule CHEMBL1651534
Route Oral Oral solution of 0.5mg given once daily for 14 days.” NCT00836082
Target FAAH “PF-04457845 has been shown to inactivate the FAAH enzyme in animals and healthy human volunteers.” NCT00981357