Drugs / cilengitide
last change Jun 2017 re-read 2 minutes ago

cilengitide

also known as EMD121974 · NSC 707544 · Cil · Cilengitida · EMD-12192

Peptide

Developed for
glioblastoma · adult glioblastoma · giant cell glioblastoma · gliosarcoma · cancer of unknown primary site · central nervous system neoplasm · childhood cerebral astrocytoma · non-small cell lung carcinoma
+60 more · optic pathway glioma · acute basophilic leukemia · acute megakaryoblastic leukemia in adult · acute myeloblastic leukemia without maturation · acute myeloid leukemia with 11q23 abnormalities · acute myeloid leukemia with minimal differentiation · adult acute monocytic leukemia · adult T-cell leukemia/lymphoma · AIDS-related primary central nervous system lymphoma · anaplastic astrocytoma · anaplastic large cell lymphoma · anaplastic oligodendroglioma · angioimmunoblastic T-cell lymphoma · benign meningioma · Burkitt lymphoma · cerebellar astrocytoma · childhood brain stem glioma · childhood central nervous system germ cell tumor · childhood cerebellar astrocytic neoplasm · childhood choroid plexus neoplasm · childhood medulloblastoma · childhood oligodendroglioma · chronic lymphocytic leukemia/small lymphocytic lymphoma · craniopharyngioma · diffuse intrinsic pontine glioma · diffuse large B-cell lymphoma · ependymoblastoma · erythroleukemia · glioma · grade II meningioma · grade III meningioma · grade III prostatic intraepithelial neoplasia · Hodgkins lymphoma · intraocular lymphoma · large-cell immunoblastic lymphoma · leukemia · lung cancer · male breast carcinoma · MALT lymphoma · mantle cell lymphoma · medulloepithelioma · melanoma · mixed glioma · mycosis fungoides and variants · myelodysplastic syndrome · myeloproliferative neoplasm · nodal marginal zone B-cell lymphoma · pediatric infratentorial ependymoma · pediatric supratentorial ependymoma · pineoblastoma · plasma cell neoplasm · precancerous condition · prostate carcinoma · sarcoma · small intestine cancer · splenic marginal zone lymphoma · squamous cell carcinoma · subependymal giant cell astrocytoma · supratentorial primitive neuroectodermal tumor · triple-negative breast carcinoma
Investigated by
National Cancer Institute (NCI) · Merck KGaA, Darmstadt, Germany · EMD Serono · Brain Tumor Trials Collaborative · Centre Oscar Lambret · European Organisation for Research and Treatment of Cancer - EORTC
+8 more · Heidelberg University · Indiana University · Institut Claudius Regaud · M.D. Anderson Cancer Center · Martin-Luther-University Halle-Wittenberg · New Approaches to Brain Tumor Therapy Consortium · Northern Sydney and Central Coast Area Health Service · University Medical Center Mannheim

Trials 29 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 113 trials
Phase 1 NCT01558687 Aug 2012 → Feb 2013 glioblastoma Merck KGaA, Darmstadt, Germany Terminated No outcome recorded
Phase 1 NCT01504165 Jan → Apr 2012 impaired renal function disease Merck KGaA, Darmstadt, Germany Completed No outcome recorded
Phase 1 NCT01276496 Dec 2010 → Mar 2015 male breast carcinoma, triple-negative breast carcinoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 1 NCT01165333 Sep 2010 → Jan 2014 diffuse intrinsic pontine glioma Centre Oscar Lambret Completed No outcome recorded
Phase 1 NCT01118676 Mar 2010 → Apr 2015 non-small cell lung carcinoma Institut Claudius Regaud Completed No outcome recorded
Phase 1 NCT00979862 Mar 2010 → May 2012 adult glioblastoma, giant cell glioblastoma, gliosarcoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 1 NCT01122888 Dec 2009 → Sep 2012 adult glioblastoma, giant cell glioblastoma, gliosarcoma National Cancer Institute (NCI) Terminated No outcome recorded
Phase 1 NCT00884598 Dec 2008 → Oct 2012 central nervous system neoplasm, lung cancer University Medical Center Mannheim Completed No outcome recorded
Phase 1 NCT00077155 Dec 2003 → Jun 2010 AIDS-related primary central nervous system lymphoma, Burkitt lymphoma, Hodgkins lymphoma, MALT lymphoma +11 National Cancer Institute (NCI) Completed No outcome recorded
Phase 1 NCT00063973 Jul 2003 → Mar 2008 benign meningioma, childhood brain stem glioma, childhood central nervous system germ cell tumor, childhood cerebellar astrocytic neoplasm +16 National Cancer Institute (NCI) Completed No outcome recorded
Phase 1/23 trials
Phase 1/2 NCT00705016 Oct 2008 → Sep 2011 squamous cell carcinoma Merck KGaA, Darmstadt, Germany Completed No outcome recorded
Phase 1/2 NCT00085254 Apr 2005 → Nov 2012 adult glioblastoma, giant cell glioblastoma, gliosarcoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 1/2 NCT00006093 Sep 2000 → Oct 2006 central nervous system neoplasm New Approaches to Brain Tumor Therapy Consortium Completed No outcome recorded
Phase 212 trials
Phase 2 NCT01782976 Jun 2013 → Jun 2017 glioblastoma M.D. Anderson Cancer Center Withdrawn No outcome recorded
Phase 2 NCT01517776 Jan 2012 → Mar 2014 glioma Martin-Luther-University Halle-Wittenberg Terminated No outcome recorded
Phase 2 NCT01124240 Nov 2009 → Nov 2012 glioblastoma Northern Sydney and Central Coast Area Health Service Unknown No outcome recorded
Phase 2 NCT00813943 Mar 2009 → Feb 2013 glioblastoma EMD Serono Completed No outcome recorded
Phase 2 NCT00842712 Feb 2009 → Jul 2013 non-small cell lung carcinoma Merck KGaA, Darmstadt, Germany Completed No outcome recorded
Phase 2 NCT00679354 Jun 2008 → Oct 2010 anaplastic astrocytoma, anaplastic oligodendroglioma, cerebellar astrocytoma, childhood cerebral astrocytoma +2 National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT00121238 Jan 2005 → Nov 2010 grade III prostatic intraepithelial neoplasia National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT00112866 Jan 2005 → Dec 2008 adult glioblastoma, giant cell glioblastoma, gliosarcoma National Cancer Institute (NCI) Terminated No outcome recorded
Phase 2 NCT00103337 Jan 2005 → Oct 2007 prostate carcinoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT00093964 Oct 2004 → Oct 2005 glioblastoma EMD Serono Completed No outcome recorded
Phase 31 trial
Phase 3 NCT00689221 Sep 2008 → Nov 2012 glioblastoma EMD Serono Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT01044225 Comparator Sep 2009 → Sep 2011 glioblastoma Bart Neyns Terminated No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 35 sources stand behind the page.

FieldValueCited text
Known as Cilengitide “Subjects will receive cilengitide monotherapy for 2 weeks (Weeks 1 and 2); thereafter, cilengitide will be given in combination with the standard treatment regimen during Weeks 3 to 36.” NCT01558687
29

NCT00842712

NCT00063973

NCT01517776

NCT00979862

NCT00813943

NCT01165333

NCT00705016

NCT00089388

NCT00884598

NCT00006093

NCT00103337

NCT01118676

NCT00085254

NCT01044225

NCT00006222

NCT01504165

NCT01122888

NCT01782976

NCT00093964

NCT00112866

NCT01124240

NCT00077155

NCT00022113

NCT00679354

NCT00689221

NCT00121238

NCT00004258

NCT00082875

NCT01276496

Known as Cil Cilengitide (Cil) will be administered at a dose of 1000 milligram (mg) as intravenous infusion twice weekly over 1 hour on Days 1 and 4.” NCT00842712
Known as Cilengitida ChEMBL registry synonym — accepted as the source's own label CHEMBL429876
Known as EMD-12192 ChEMBL registry synonym — accepted as the source's own label CHEMBL429876
Known as EMD121974 “A Multi-center, Open-label, Randomized, Controlled Phase I Trial to Investigate the Effects of Cilengitide (EMD 121974) Using Dynamic MR and FET-PET Imaging as a...” NCT01558687
6

“This multi-institutional phase I trial was designed to determine the maximum-tolerated dose (MTD) of cilengitide (EMD 121974) and to evaluate the use of perfusion magnetic...” PMID 17470857 May 2007

“Cilengitide (EMD121974) in Combination With Whole Brain Radiotherapy in Patients With Brain Metastases From Lung Cancer” NCT00884598

“Cilengitide (EMD 121974) (IND# 59073) in Recurrent or Progressive and Refractory Childhood High-Grade Glioma” NCT00679354

“Cilengitide (EMD121974; Merck KgaA, Darmstadt, Germany), a cyclic pentapeptide containing the sequence RGD” NCT01165333

“Cilengitide (EMD 121974) may stop the growth of cancer cells by stopping blood flow to the cancer” NCT00077155

“Patients receive cilengitide (EMD 121974) IV over 1 hour twice weekly.” NCT00063973

Known as NSC 707544 “Phase II study of cilengitide (EMD 121974, NSC 707544) in patients with non-metastatic castration resistant prostate cancer, NCI-6735.” PMID 21049281 Nov 2010
1

“A Phase 2 Study of EMD 121974 (Cilengitide, NSC 707544) in Patients With Metastatic Melanoma” NCT00082875

Action Inhibit “Cilengitide is a selective integrin inhibitor that is well tolerated and has demonstrated biologic activity in patients with recurrent malignant glioma.” PMID 22517399 Apr 2012
Modality Peptide “Randomized phase II study of cilengitide, an integrin-targeting arginine-glycine-aspartic acid peptide, in recurrent glioblastoma multiforme.” PMID 18981465 Nov 2008
Route Intravenous “administered as a twice weekly intravenous infusion” PMID 17470857 May 2007