Drugs / Trebananib
last change Dec 2024 re-read 2 minutes ago

Trebananib

also known as AMG 386 · Amgen 386

Peptide targets ANGPT1, ANGPT2 via inhibition

Developed for
cancer · fallopian tube cancer · ovarian cancer · primary peritoneal carcinoma · angiosarcoma · carcinoma · fallopian tube carcinoma · female breast carcinoma
+40 more · neoplasm · ovarian carcinoma · renal cell carcinoma · acute erythroid leukemia · acute megakaryoblastic leukemia in adult · acute myeloblastic leukemia with maturation · acute myeloblastic leukemia without maturation · acute myeloid leukemia with 11q23 abnormalities · acute myeloid leukemia with minimal differentiation · acute myeloid leukemia with t(8;21)(q22;q22) translocation · acute myeloid leukemia, del(5q31-q32) · acute myeloid leukemia, inv(16)(p13.1;q22) · acute myeloid leukemia, t(16;16)(p13.1;q22) · acute myelomonocytic leukemia M4 · adult acute monocytic leukemia · cancer or benign tumor · central nervous system neoplasm · clear cell renal carcinoma · colorectal cancer · digestive system cancer · digestive system neuroendocrine tumor, grade 1/2 · endometrial adenosquamous carcinoma · endometrial clear cell adenocarcinoma · endometrial serous adenocarcinoma · endometrioid adenocarcinoma · endometrioid stromal sarcoma · giant cell glioblastoma · glioblastoma · gliosarcoma · hepatocellular carcinoma · Her2-receptor negative breast cancer · lung carcinoid tumor · non-small cell lung carcinoma · oligodendroglioma · peritoneum cancer · prostate cancer · sarcomatoid renal cell carcinoma · urothelial carcinoma · uterine corpus sarcoma · breast cancer
Investigated by
Amgen · National Cancer Institute (NCI) · Dana-Farber Cancer Institute · Austin Health · Gynecologic Oncology Group · Merck Sharp & Dohme LLC
+5 more · NRG Oncology · QuantumLeap Healthcare Collaborative · Roswell Park Cancer Institute · Takeda · University of Colorado, Denver

Trials 30 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 112 trials
Phase 1 NCT03239145 May 2018 → Dec 2024 cancer or benign tumor Dana-Farber Cancer Institute Completed No outcome recorded
Phase 1 NCT01992341 Jul 2012 → Aug 2013 cancer Amgen Completed No outcome recorded
Phase 1 NCT01548482 Mar 2012 → Jan 2014 digestive system neuroendocrine tumor, grade 1/2, lung carcinoid tumor, renal cell carcinoma, uterine corpus sarcoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 1 NCT01538095 Feb 2012 → Apr 2016 central nervous system neoplasm National Cancer Institute (NCI) Completed No outcome recorded
Phase 1 NCT01555268 Oct 2011 → Sep 2013 acute erythroid leukemia, acute megakaryoblastic leukemia in adult, acute myeloblastic leukemia with maturation, acute myeloblastic leukemia without maturation +8 Roswell Park Cancer Institute Completed No outcome recorded
Phase 1 NCT01331941 Sep 2011 → Feb 2013 cancer, impaired renal function disease Amgen Completed No outcome recorded
Phase 1 NCT01253681 Nov 2010 → Oct 2012 carcinoma, fallopian tube cancer, ovarian cancer, peritoneum cancer Amgen Completed No outcome recorded
Phase 1 NCT02525536 Jun 2009 → May 2014 neoplasm Takeda Completed No outcome recorded
Phase 1 NCT00807859 Mar 2009 → Feb 2014 female breast carcinoma, metastatic malignant neoplasm Amgen Completed No outcome recorded
Phase 1 NCT00770536 Jan 2009 → Jan 2012 carcinoma, fallopian tube cancer, metastatic neoplasm, ovarian cancer Amgen Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT01666977 Aug 2012 → Nov 2015 non-small cell lung carcinoma Amgen Completed No outcome recorded
Phase 1/2 NCT01290263 Dec 2010 → Jul 2015 glioblastoma Dana-Farber Cancer Institute Completed No outcome recorded
Phase 214 trials
Phase 2 NCT01907308 Feb → Apr 2014 urothelial carcinoma University of Colorado, Denver Withdrawn No outcome recorded
Phase 2 NCT01664182 Aug 2012 → Dec 2020 sarcomatoid renal cell carcinoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT01623869 Jul 2012 → Sep 2014 angiosarcoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT01609790 Jun 2012 → Oct 2015 giant cell glioblastoma, gliosarcoma, oligodendroglioma National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT01553188 Feb 2012 → Apr 2017 prostate cancer National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT01210222 Jun 2011 → Jul 2016 endometrial adenosquamous carcinoma, endometrial clear cell adenocarcinoma, endometrial serous adenocarcinoma, endometrioid adenocarcinoma +1 Gynecologic Oncology Group Completed No outcome recorded
Phase 2 NCT01249521 Nov 2010 → Nov 2011 colorectal cancer Austin Health Unknown No outcome recorded
Phase 2 NCT01042379 Mar 2010 → Dec 2030 expected HER2 positive breast carcinoma, angiosarcoma, female breast carcinoma, hormone receptor-positive breast cancer +1 QuantumLeap Healthcare Collaborative Recruiting No outcome recorded
Phase 2 NCT00872014 Aug 2009 → Oct 2011 hepatocellular carcinoma Amgen Completed No outcome recorded
Phase 2 NCT00853372 May 2009 → Aug 2011 renal cell carcinoma Amgen Completed No outcome recorded
Phase 32 trials
Phase 3 NCT01281254 Apr 2011 → Aug 2014 fallopian tube cancer, ovarian carcinoma, primary peritoneal carcinoma Amgen Terminated No outcome recorded
Phase 3 NCT01204749 Nov 2010 → Mar 2013 fallopian tube carcinoma, ovarian cancer, primary peritoneal carcinoma Amgen Completed No outcome recorded
Also used as a comparator or background therapy in 2 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 21 trial
Phase 2 NCT00752570 Comparator Nov 2008 → Sep 2010 colon carcinoma, metastatic malignant neoplasm, rectal cancer Amgen Completed No outcome recorded
Phase 31 trial
Phase 3 NCT01493505 Comparator Jan 2012 → Mar 2016 fallopian tube cancer, ovarian cancer, peritoneum cancer Amgen Terminated No outcome recorded

Press releases naming this drug 1 release

DateIssuerRelease
2014-11-05 Takeda Takeda Announces Topline Secondary Endpoint Results from the Phase 3 TRINOVA-1 Trial of Trebananib (AMG 386) for Recurrent Ovarian Cancer takeda.com

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 35 sources stand behind the page.

FieldValueCited text
Known as Trebananib Trebananib (AMG 386) plus weekly paclitaxel with or without bevacizumab as first-line therapy for HER2-negative locally recurrent or metastatic breast cancer: A phase 2...” PMID 25747197 Mar 2015
13

“A randomised, double-blind, placebo-controlled phase 2 study of trebananib (AMG 386) in combination with FOLFIRI in patients with previously treated metastatic colorectal carcinoma.” PMID 23361051 Jan 2013

“A phase 1b, open-label study of trebananib in combination with paclitaxel and” PMID 25037684 Jul 2014

“AMG 386 (Trebananib) in Ovarian Cancer (TRINOVA-2)” NCT01281254

NCT01210222

NCT03239145

NCT01623869

NCT01538095

NCT01664182

NCT02525536

NCT00853372

NCT01609790

NCT01555268

NCT01548482

Known as AMG 386 “To estimate the proportion of patients with persistent or recurrent endometrial cancer, who survive progression-free for at least 6 months and the proportion of patients who...” NCT01210222
22

“Trebananib (AMG 386) plus weekly paclitaxel with or without bevacizumab as first-line therapy for HER2-negative locally recurrent or metastatic breast cancer: A phase 2...” PMID 25747197 Mar 2015

“A randomised, double-blind, placebo-controlled phase 2 study of trebananib (AMG 386) in combination with FOLFIRI in patients with previously treated metastatic colorectal carcinoma.” PMID 23361051 Jan 2013

“The drug being tested in this study is called trebananib (AMG 386).” NCT02525536

AMG 386 (Trebananib) in Ovarian Cancer (TRINOVA-2)” NCT01281254

NCT00102830

NCT01493505

NCT00807859

NCT01204749

NCT00770536

NCT01907308

NCT00479817

NCT01253681

NCT00861419

NCT01042379

NCT01553188

NCT00583674

NCT00872014

NCT01992341

NCT00467025

NCT01331941

NCT01249521

NCT01666977

Known as Amgen 386 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01290263
Action Inhibit “neutralizes the interaction of angiopoietin-1 and angiopoietin-2 with Tie2” PMID 22692704 Jun 2012
2

“Angiopoietin-1 inhibitor” CHEMBL2108568

“Angiopoietin-2 inhibitor” CHEMBL2108568

Modality Peptide “AMG 386, a peptibody (a peptide Fc fusion)” PMID 22692704 Jun 2012
Route Intravenous “after intravenous administration” NCT00102830
Target ANGPT1 “Angiopoietin-1 inhibitor” CHEMBL2108568
Target ANGPT2 “Angiopoietin-2 inhibitor” CHEMBL2108568