Drugs / Nelarabine
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Nelarabine

also known as 506U78 · 506U · Arranon · Atriance · Attriance · GW-506U78 · Nelarabina · Nelzarabine · +3 more

Small molecule

Developed for
leukemia · T-cell acute lymphoblastic leukemia · T-lymphoblastic lymphoma · acute lymphoblastic leukemia · adult T-cell leukemia/lymphoma · angioimmunoblastic T-cell lymphoma · lymphoma · mycosis fungoides and variants
+17 more · T-cell childhood acute lymphocytic leukemia · acute leukemia of ambiguous lineage · anaplastic large cell lymphoma · chronic lymphocytic leukemia/small lymphocytic lymphoma · lymphoid leukemia · MALT lymphoma · myelodysplastic syndrome · myeloproliferative neoplasm · nodal marginal zone B-cell lymphoma · plasma cell neoplasm · primary cutaneous T-cell non-Hodgkin lymphoma · small intestine lymphoma · splenic marginal zone lymphoma · T lymphoblastic leukemia/lymphoma · T-cell adult acute lymphocytic leukemia · T-cell leukemia · Waldenstrom macroglobulinemia
Investigated by
National Cancer Institute (NCI) · GlaxoSmithKline · Goethe University · M.D. Anderson Cancer Center · SWOG Cancer Research Network · Alliance for Clinical Trials in Oncology
+13 more · Assistance Publique - Hôpitaux de Paris · Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · Children's Cancer Group · National Institutes of Health (NIH) · Novartis · Novartis Pharmaceuticals · Spectrum Pharmaceuticals, Inc · St. Jude Children's Research Hospital · The Leukemia and Lymphoma Society · Therapeutic Advances in Childhood Leukemia Consortium · University College, London · University of Washington · Washington University School of Medicine

Regulatory milestones approvals, filings & regulatory actions · 3 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansion US (FDA) ARRANON 2019-07-31 fda.gov
Approved EU (EMA) Atriance 2007-08-22 europa.eu
Approved US (FDA) ARRANON 2005-10-28 fda.gov

Trials 21 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01094860 Jun 2010 → Aug 2018 leukemia M.D. Anderson Cancer Center Completed No outcome recorded
Phase 1 NCT00004239 Dec 1999 → Jan 2002 leukemia, myelodysplastic syndrome, myeloproliferative neoplasm, plasma cell neoplasm Alliance for Clinical Trials in Oncology Terminated No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00981799 Jun 2010 → Nov 2015 T-cell acute lymphoblastic leukemia, T-lymphoblastic lymphoma Therapeutic Advances in Childhood Leukemia Consortium Terminated No outcome recorded
Phase 212 trials
Phase 2 NCT02763384 Dec 2016 → Feb 2022 T-cell acute lymphoblastic leukemia, T-lymphoblastic lymphoma Washington University School of Medicine Terminated No outcome recorded
Phase 2 NCT02518750 Nov 2016 → Mar 2018 T-cell leukemia, acute lymphoblastic leukemia St. Jude Children's Research Hospital Terminated No outcome recorded
Phase 2 NCT02619630 Dec 2015 → Dec 2020 T-cell adult acute lymphocytic leukemia Assistance Publique - Hôpitaux de Paris Unknown No outcome recorded
Phase 2 NCT00501826 Jul 2007 → Oct 2026 expected T-cell acute lymphoblastic leukemia, T-lymphoblastic lymphoma M.D. Anderson Cancer Center Recruiting No outcome recorded
Phase 2 NCT00684619 Jun 2003 → Dec 2008 T lymphoblastic leukemia/lymphoma Goethe University Completed No outcome recorded
Phase 2 NCT00006020 Jul 2000 → Jun 2004 leukemia SWOG Cancer Research Network Completed No outcome recorded
Phase 2 NCT00005080 May 2000 → Jan 2006 adult T-cell leukemia/lymphoma, anaplastic large cell lymphoma, angioimmunoblastic T-cell lymphoma, mycosis fungoides and variants +1 National Cancer Institute (NCI) Completed No outcome recorded
Phase 2 NCT00005982 Apr 2000 → Jul 2004 mycosis fungoides and variants, primary cutaneous T-cell non-Hodgkin lymphoma National Cancer Institute (NCI) Terminated No outcome recorded
Phase 2 NCT00005950 Apr 2000 → Oct 2004 MALT lymphoma, Waldenstrom macroglobulinemia, adult T-cell leukemia/lymphoma, angioimmunoblastic T-cell lymphoma +3 National Cancer Institute (NCI) Terminated No outcome recorded
Phase 2 NCT00003635 Jan 1999 → Mar 2004 lymphoid leukemia GlaxoSmithKline Completed No outcome recorded
Phase 32 trials
Phase 3 NCT06434467 May 2024 → Dec 2025 T-cell acute lymphoblastic leukemia, T-lymphoblastic lymphoma Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Unknown No outcome recorded
Phase 3 NCT02881086 Aug 2016 → Dec 2024 acute lymphoblastic leukemia, lymphoblastic lymphoma Goethe University Completed No outcome recorded
Phase not applicable3 trials
NCT02551718 Sep 2015 → Jun 2020 acute leukemia of ambiguous lineage, acute lymphoblastic leukemia University of Washington Completed No outcome recorded
NCT00016302 Apr 2001 → Jul 2007 T-cell childhood acute lymphocytic leukemia National Cancer Institute (NCI) Completed No outcome recorded
NCT00003837 Sep 1999 → Nov 2007 leukemia, lymphoma National Cancer Institute (NCI) Completed No outcome recorded
Phase not stated1 trial
NCT01085617 Dec 2010 → Feb 2025 leukemia, mouth disorder, mucositis University College, London Completed No outcome recorded
Also used as a comparator or background therapy in 10 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT03328104 Background Jul 2018 → Jun 2023 T-lymphoblastic lymphoma Emory University Completed No outcome recorded
Phase 1 NCT00406757 Comparator Aug 2006 → Jul 2009 T lymphoblastic leukemia/lymphoma GlaxoSmithKline Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT07294677 Background Mar 2026 → Mar 2032 expected leukemia, lymphoma University of Chicago Recruiting No outcome recorded
Phase 1/2 NCT03808610 Background Apr 2019 → May 2026 B-cell acute lymphoblastic leukemia, T-cell acute lymphoblastic leukemia M.D. Anderson Cancer Center Terminated No outcome recorded
Phase 22 trials
Phase 2 NCT06390319 Background Dec 2024 → Dec 2027 expected T-cell acute lymphoblastic leukemia, T-cell non-Hodgkin lymphoma, mixed phenotype acute leukemia St. Jude Children's Research Hospital Recruiting No outcome recorded
Phase 2 NCT06210750 Background Aug 2024 → Sep 2026 T-cell acute lymphoblastic leukemia, T-lymphoblastic lymphoma National Cancer Institute (NCI) Withdrawn No outcome recorded
Phase 2/32 trials
Phase 2/3 NCT07072585 Background Aug 2026 → Sep 2035 expected T-cell acute lymphoblastic leukemia, T-lymphoblastic lymphoma Children's Oncology Group Not yet recruiting No outcome recorded
Phase 2/3 NCT03117751 Background Mar 2017 → Sep 2026 expected lymphoblastic leukemia, acute, with lymphomatous features St. Jude Children's Research Hospital Active not recruiting No outcome recorded
Phase 32 trials
Phase 3 NCT03020030 Background Mar 2017 → Nov 2026 expected childhood acute lymphoblastic leukemia Dana-Farber Cancer Institute Active not recruiting No outcome recorded
Phase 3 NCT00408005 Comparator Jan 2007 → Sep 2017 T-cell acute lymphoblastic leukemia, T-lymphoblastic lymphoma National Cancer Institute (NCI) Completed No outcome recorded

Evidence & citations 14 cited values

Every value below carries the sentence it was read from. 33 sources stand behind the page.

FieldValueCited text
Known as nelarabine “Mitoxantrone Nelarabine Nilotinib” NCT02551718
29

NCT01085617

NCT00016302

NCT07072585

NCT00003545

NCT02518750

NCT02763384

NCT06210750

NCT00684619

NCT03117751

NCT00005080

NCT02619630

NCT00005982

NCT03808610

NCT01094860

NCT00981799

NCT03020030

NCT00003635

NCT07294677

NCT06434467

NCT00501826

NCT00408005

NCT00005950

NCT00002970

NCT02881086

NCT00406757

NCT00003837

NCT03328104

NCT00006020

NCT06390319

Known as 506U ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as 506U78 “Nelarabine (506U78) is a soluble pro-drug of 9-beta-D-arabinofuranosylguanine (ara-G), a deoxyguanosine derivative.” PMID 17344466 Mar 2007
2

“Clinical Evaluation of Nelarabine (506U78)in Japanese Patients With Leukemia or Lymphoma” NCT00406757

NCT00004239

Known as Arranon ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as Atriance ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as Attriance ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as GW-506U78 ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as Nelarabina ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as Nelzarabine ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as NSC #686673 “Compound 506U78 (NSC #686673)” NCT00004239
Known as NSC-755985 ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Known as NSC-759876 ChEMBL registry synonym — accepted as the source's own label CHEMBL1201112
Modality Small molecule “Nelarabine (506U78) is a soluble pro-drug of 9-beta-D-arabinofuranosylguanine (ara-G), a deoxyguanosine derivative.” PMID 17344466 Mar 2007
Route Intravenous “Given IV” NCT00002970