Drugs / Ivacaftor

Regulatory milestones approvals, filings & regulatory actions · 13 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (11) US (FDA) KALYDECO 2014-02-21 – 2025-05-22 fda.gov
Approved EU (EMA) Kalydeco 2012-07-23 europa.eu
Approved US (FDA) KALYDECO 2012-01-31 fda.gov

Trials 93 · started per year

today
US approved 2012
EU approved 2012
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200720082009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 02 trials
Phase 0 NCT03439865 May 2019 → Apr 2027 expected chronic rhinosinusitis University of Alabama at Birmingham Recruiting No outcome recorded
Phase 0 NCT02135432 May → Oct 2015 chronic obstructive pulmonary disease University of Alabama at Birmingham Completed No outcome recorded
Phase 111 trials
Phase 1 NCT02015507 Jan → Feb 2014 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01899105 Jul → Aug 2013 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01888393 Jun → Nov 2013 Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01910415 Jun 2013 → Mar 2014 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01768663 Jan → Sep 2013 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01216046 Oct 2010 → May 2011 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01208285 Sep → Dec 2010 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01153542 Jun → Aug 2010 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01060566 Feb → Mar 2010 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT01018368 Nov 2009 → Mar 2010 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 217 trials
Phase 2 NCT04581408 Jun 2021 → Apr 2025 long QT syndrome Istituto Auxologico Italiano Completed No outcome recorded
Phase 2 NCT04135495 Nov 2019 → Oct 2022 cystic fibrosis Eloxx Pharmaceuticals, Inc. Completed No outcome recorded
Phase 2 NCT04126473 Nov 2019 → Apr 2022 cystic fibrosis Eloxx Pharmaceuticals, Inc. Completed No outcome recorded
Phase 2 NCT03506061 Sep 2019 → Feb 2024 cystic fibrosis Emory University Completed No outcome recorded
Phase 2 NCT03625466 Aug 2018 → Oct 2020 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 2 NCT03061331 Jan → Sep 2017 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 2 NCT02730208 Sep 2016 → Jul 2018 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 2 NCT02871778 Aug 2016 → Nov 2018 primary ciliary dyskinesia Parion Sciences Completed No outcome recorded
Phase 2 NCT02508207 Feb 2016 → Jun 2017 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 2 NCT02070744 Mar 2014 → May 2016 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 346 trials
Phase 3 NCT06460506 Nov 2024 → Sep 2027 expected cystic fibrosis Vertex Pharmaceuticals Incorporated Active not recruiting No outcome recorded
Phase 3 NCT05331183 Nov 2022 → Apr 2027 expected cystic fibrosis Vertex Pharmaceuticals Incorporated Active not recruiting No outcome recorded
Phase 3 NCT05274269 May 2022 → Jul 2023 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT05153317 Jan 2022 → Jan 2026 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT05111145 Jan → Dec 2022 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT04969224 Oct 2021 → Jul 2022 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT04545515 Jan 2021 → Mar 2023 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT04362761 May 2020 → Dec 2022 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT04235140 Feb 2020 → Aug 2023 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT04058366 Dec 2019 → Dec 2022 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 48 trials
Phase 4 NCT07148739 Jun 2025 → Dec 2030 expected cystic fibrosis Arkansas Children's Hospital Research Institute Recruiting No outcome recorded
Phase 4 NCT05743946 Apr 2023 → Dec 2025 bronchiectasis Emory University Completed No outcome recorded
Phase 4 NCT04840862 May 2022 → May 2024 University of Southern California Completed No outcome recorded
Phase 4 NCT03251911 Jan 2020 → Feb 2022 chronic bronchitis University of Alabama at Birmingham Withdrawn No outcome recorded
Phase 4 NCT03624101 Dec 2018 → Oct 2019 cystic fibrosis University of Alabama at Birmingham Terminated No outcome recorded
Phase 4 NCT03956589 Oct 2018 → Apr 2020 cystic fibrosis University Hospital, Antwerp Terminated No outcome recorded
Phase 4 NCT03256799 Mar → Jul 2017 cystic fibrosis University of Alabama at Birmingham Completed No outcome recorded
Phase 4 NCT02875366 Sep 2016 → Sep 2017 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase not applicable6 trials
NCT04580368 May 2021 → Dec 2028 expected cystic fibrosis Children's Hospital Medical Center, Cincinnati Recruiting No outcome recorded
NCT04415268 Jun 2020 → Jan 2021 cystic fibrosis Universidad Europea de Madrid Withdrawn No outcome recorded
NCT02653027 Jan → Feb 2018 cystic fibrosis, diabetes mellitus Massachusetts General Hospital Withdrawn No outcome recorded
NCT02858843 Aug 2016 → May 2018 cystic fibrosis, diabetes mellitus Massachusetts General Hospital Terminated No outcome recorded
NCT02310789 Jul 2015 → Aug 2016 cystic fibrosis Richard Barry Moss Completed No outcome recorded
NCT01784419 Oct 2013 → Dec 2015 cystic fibrosis University of California, San Francisco Completed No outcome recorded
Phase not stated3 trials
NCT04058210 cystic fibrosis Vertex Pharmaceuticals Incorporated Approved for marketing No outcome recorded
NCT03278314 cystic fibrosis Vertex Pharmaceuticals Incorporated Approved for marketing No outcome recorded
NCT01381289 cystic fibrosis Vertex Pharmaceuticals Incorporated Approved for marketing No outcome recorded
Also used as a comparator or background therapy in 18 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT03029455 Background Nov 2016 → Aug 2017 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT02599792 Comparator Nov 2015 → Apr 2016 Concert Pharmaceuticals Completed No outcome recorded
Phase 1 NCT02392702 Comparator Mar → Jun 2015 Concert Pharmaceuticals Completed No outcome recorded
Phase 26 trials
Phase 2 NCT06237335 Background Feb 2024 → Aug 2026 overdue cystic fibrosis ReCode Therapeutics Recruiting No outcome recorded
Phase 2 NCT04066751 Comparator Dec 2021 → Oct 2024 chronic obstructive pulmonary disease University of Alabama at Birmingham Withdrawn No outcome recorded
Phase 2 NCT04006873 Comparator Sep 2019 → Oct 2020 cystic fibrosis Nottingham University Hospitals NHS Trust Completed No outcome recorded
Phase 2 NCT03085485 Comparator Mar 2017 → Sep 2022 chronic bronchitis University of Alabama at Birmingham Completed No outcome recorded
Phase 2 NCT02951195 Background Nov 2016 → Jan 2018 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 36 trials
Phase 3 NCT05033080 Comparator Sep 2021 → May 2023 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT04183790 Background Feb 2020 → Feb 2024 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT04058353 Background Aug 2019 → Jun 2020 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT03525548 Background Aug → Dec 2018 cystic fibrosis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 3 NCT03447262 Background Jul 2018 → Sep 2020 cystic fibrosis Vertex Pharmaceuticals Incorporated Terminated No outcome recorded
Phase 42 trials
Phase 4 NCT02823470 Background Jun 2016 → Aug 2017 cystic fibrosis Vertex Pharmaceuticals Incorporated Terminated No outcome recorded
Phase 4 NCT01937325 Comparator Feb → Dec 2014 cystic fibrosis The Alfred Unknown No outcome recorded
Phase not applicable1 trial
NCT03894657 Background Dec 2019 → Nov 2021 cystic fibrosis Assistance Publique - Hôpitaux de Paris Completed No outcome recorded

Press releases naming this drug 161 releases

DateIssuerRelease
2025-04-07 Vertex Pharmaceuticals Incorporated European Commission Approves Expanded Label for KAFTRIO® in Combination With Ivacaftor for People With Cystic Fibrosis vrtx.com
2025-02-28 Vertex Pharmaceuticals Incorporated Vertex Receives CHMP Positive Opinion for Expanded Label for KAFTRIO® in Combination With Ivacaftor for People With Cystic Fibrosis to Include Rare Mutations vrtx.com
2024-12-20 Vertex Pharmaceuticals Incorporated Vertex Announces U.S. FDA Approval for TRIKAFTA (elexacaftor/tezacaftor/ivacaftor and ivacaftor) to Include Additional Non-F508del TRIKAFTA-Responsive Variants vrtx.com
2024-04-26 Vertex Pharmaceuticals Incorporated Vertex Announces European Commission Approval for KALYDECO® to Treat Infants With Cystic Fibrosis Ages 1 Month and Older vrtx.com
2024-02-23 Vertex Pharmaceuticals Incorporated Vertex Receives CHMP Positive Opinion for KALYDECO® for the Treatment of Infants With Cystic Fibrosis Ages 1 Month and Older vrtx.com
2023-11-24 Vertex Pharmaceuticals Incorporated Vertex Announces European Medicines Agency Validation for Marketing Authorization Application Extension for KAFTRIO® in Combination With Ivacaftor to Include People With Cystic Fibrosis and Responsive Rare Mutations vrtx.com
2023-11-23 Vertex Pharmaceuticals Incorporated European Commission Approves KAFTRIO® in Combination With Ivacaftor for the Treatment of Children With Cystic Fibrosis Ages 2 Through 5 vrtx.com
2023-09-15 Vertex Pharmaceuticals Incorporated Vertex Receives CHMP Positive Opinion for KAFTRIO® (ivacaftor/tezacaftor/elexacaftor) in Combination With Ivacaftor for Children With Cystic Fibrosis Ages 2 Through 5 vrtx.com
2023-07-05 Vertex Pharmaceuticals Incorporated European Commission Approves ORKAMBI® (lumacaftor/ivacaftor) for the Treatment of Children With Cystic Fibrosis Ages 1 to <2 Years Old vrtx.com
2023-05-03 Vertex Pharmaceuticals Incorporated Vertex Announces U.S. FDA Approval for KALYDECO® (ivacaftor) to Treat Eligible Infants With CF Ages 1 Month and Older vrtx.com
2023-04-27 Vertex Pharmaceuticals Incorporated Vertex Receives CHMP Positive Opinion for ORKAMBI® (lumacaftor/ivacaftor) in Children With Cystic Fibrosis Ages 1 to <2 Years Old vrtx.com
2023-04-26 Vertex Pharmaceuticals Incorporated Vertex Announces U.S. FDA Approval for TRIKAFTA® (elexacaftor/tezacaftor/ivacaftor and ivacaftor) in Children With Cystic Fibrosis Ages 2 Through 5 With Certain Mutations vrtx.com
Show all 161 releases opens the full record — a long page

Evidence & citations 11 cited values

Every value below carries the sentence it was read from. 116 sources stand behind the page.

FieldValueCited text
Known as ivacaftor “received weight-based and age-based doses of oral lumacaftor-ivacaftor: children weighing less than 14 kg and aged younger than 6 years at study 116 screening received...” PMID 33965000 May 2021
96

“This study evaluated the long-term safety, efficacy, and pharmacodynamics of elexacaftor (ELX, VX-445) in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in...” NCT04058366

“This study will evaluate the efficacy, safety and pharmacodynamics of elexacaftor (ELX, VX-445) in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects...” NCT04058353

“The purpose of this program is to provide elexacaftor(ELX, VX-445)/tezacaftor(TEZ)/ivacaftor(IVA) combination therapy to CF patients in critical need who are 12 years of age...” NCT04058210

“Following a run-in period of 4 weeks with Tezacaftor (TEZ)/Ivacaftor (IVA), participants received TEZ 100 milligram (mg)/IVA 150 mg as fixed-dose combination (FDC) tablet in...” NCT03460990

“This study will evaluate the pharmacokinetics (PK), safety, tolerability, efficacy, and pharmacodynamic effect of VX-659, tezacaftor (TEZ), and ivacaftor (IVA) when dosed in...” NCT03633526

“This is a Phase 2, randomized, double blind, placebo and active-controlled, parallel group, multicenter study designed to evaluate the safety and tolerability of VX-152 in...” NCT02951195

“The CFTR modulating drugs that are currently FDA approved and will be tested in this study include ivacaftor and the combination drugs orkambi (ivacaftor/lumacaftor), symdeko...” NCT04580368

“This study will evaluate the long-term safety and tolerability of VX-659 in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects with cystic fibrosis...” NCT03447262

“A Phase 3, Double-blind, Parallel-group Study to Evaluate the Efficacy and Safety of Tezacaftor in Combination With Ivacaftor in Subjects Aged 6 Through 11 Years With Cystic...” NCT03559062

“This study will evaluate the efficacy of VX-659 in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects with cystic fibrosis (CF) who are heterozygous...” NCT03447249

“This study will evaluate the efficacy, safety, and pharmacodynamics of elexacaftor (ELX, VX-445) in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in...” NCT04105972

“Participants will take Trikafta which is a combination tablet comprised of 100 milligrams (mg) of elexacaftor, 50 mg of tezacaftor and 75 mg of ivacaftor (2 tablets taken in...” NCT03506061

“After a 4-week tezacaftor plus ivacaftor run-in period, participants were randomly assigned (1:1) to 4 weeks of elexacaftor 200 mg orally once daily plus tezacaftor 100 mg...” PMID 31679946 Oct 2019

“Rationale: Elexacaftor (ELX)/tezacaftor (TEZ)/ivacaftor (IVA) was shown to be safe and efficacious in children 6 through 11 years of age with cystic fibrosis (CF) and at least...” PMID 40454869 Oct 2025

“The purpose of this study is to evaluate the long term safety, tolerability, efficacy and pharmacodynamics of elexacaftor (ELX)/tezacaftor (TEZ)/ivacaftor (IVA) in CF...” NCT05153317

“Participants will be given elexacaftor 100 mg/tezacaftor 50 mg/ivacaftor 75 mg (two pills once daily in the morning) and ivacaftor 150 mg (once daily in the evening), as the...” NCT05743946

“Over 120 weeks (initial study period and follow-up), systolic blood pressure rose by 5.1 mmHg and diastolic blood pressure by 4.1 mmHg with twice-daily 400 mg...” PMID 37983082 Nov 2023

“elexacaftor (200 mg once daily), tezacaftor (100 mg once daily), and ivacaftor (150 mg once every 12 h) as two fixed-dose combination tablets in the morning and one ivacaftor...” PMID 39756424 Jan 2025

“This study evaluated the long-term safety and tolerability of elexacaftor (ELX), tezacaftor (TEZ), and ivacaftor (IVA) triple combination (TC) treatment in participants with...” NCT04043806

“the mean increase in CFQ scores with twice-daily tezacaftor (100 mg) and ivacaftor (150 mg) was approximately five points (95% CI 3.20 to 7.00; 504 participants;...” PMID 33331662 Dec 2020

“Long-Term Impact of Lumacaftor/Ivacaftor Treatment on Cystic Fibrosis Disease Progression in Children 2-5 Years of Age Homozygous for F508del-CFTR: A Phase 2, Open-Label Clinical Trial.” PMID 39173175 Nov 2024

“Participants weighing less than (\<)40 kilograms (kg) at Day 1 received tezacaftor (TEZ) 50 milligrams (mg) once daily (qd)/ivacaftor (IVA) 75 mg every 12 hours (q12h)” NCT03537651

“The purpose of the study is to evaluate the long-term safety, tolerability, efficacy, and pharmacodynamics (PD) of elexacaftor (ELX)/tezacaftor (TEZ)/ivacaftor (IVA).” NCT06460506

“This study will evaluate the effects of elexacaftor/tezacaftor/ivacaftor (ELX/TEZ/IVA) on cough and physical activity using wearable technology in CF participants.” NCT04969224

“A Phase 3 Open-Label Study of Elexacaftor/Tezacaftor/Ivacaftor in Children 6 through 11 Years of Age with Cystic Fibrosis and at Least One F508del Allele.” PMID 33734030 Jun 2021

“Orkambi® is a combination of Ivacaftor (a CFTR channel potentiator) and Lumacaftor (a corrector partially rescuing the traffic of mutated CFTR).” NCT03894657

“Infants received 25 mg or 50 mg ivacaftor every 12 hours on the basis of age and weight for 4 days in part A and 24 weeks in part B.” PMID 33023304 Mar 2021

“Study to Evaluate Elexacaftor/Tezacaftor/Ivacaftor (ELX/TEZ/IVA) Long-term Safety and Efficacy in Subjects Without F508del” NCT05331183

“Lumacaftor (LUM) 200 mg every 12 hours (q12h)/ivacaftor (IVA) 250 mg q12h (for 6 through 11 years of age).” NCT02544451

“Trikafta (Elexacaftor \[ELX\], Tezacaftor \[TEZ\], Ivacaftor\[IVA\]) is contraindicated” NCT04840862

“Standard of care: Lumacaftor with Ivacaftor or Tezacaftor combined with Ivacaftor.” NCT04415268

“Lumacaftor/ivacaftor in people with cystic fibrosis with an A455E-CFTR mutation.” PMID 33249003 Nov 2020

“Children received lumacaftor 100 mg and ivacaftor 125 mg” PMID 30686767 Jan 2019

“Product ORKAMBI (Lumacaftor/ Ivacaftor) on Lung Function” NCT03956589

ivacaftor 150 mg once every 12 h for up to 96 weeks” PMID 33581080 Feb 2021

“elexacaftor (ELX)/tezacaftor (TEZ)/ivacaftor (IVA)” NCT05111145

“lumacaftor/ivacaftorNCT02823470

“Lumacaftor/IvacaftorNCT02875366

ivacaftorNCT04362761

ivacaftorNCT05274269

NCT03251911

NCT01614470

NCT02508207

NCT01946412

NCT01614457

NCT01910415

NCT01768663

NCT02934698

NCT02858843

NCT03150719

NCT01707290

NCT07148739

NCT00909727

NCT02310789

NCT03278314

NCT01705145

NCT01784419

NCT02390219

NCT06237335

NCT02412111

NCT03068312

NCT03624101

NCT01262352

NCT02015507

NCT01937325

NCT00953706

NCT04066751

NCT02653027

NCT04126473

NCT02135432

NCT01685801

NCT02070744

NCT01897233

NCT01888393

NCT04581408

NCT01117012

NCT02347657

NCT03439865

NCT00457821

NCT03256799

NCT04006873

NCT00909532

NCT02742519

NCT03085485

NCT03029455

NCT01931839

NCT02730208

NCT01899105

NCT01807949

NCT01807923

NCT02871778

NCT02516410

NCT01531673

NCT01225211

NCT04135495

NCT02392234

Known as IVA “This study evaluated the long-term safety, efficacy, and pharmacodynamics of elexacaftor (ELX, VX-445) in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in...” NCT04058366
26

“This study will evaluate the efficacy, safety and pharmacodynamics of elexacaftor (ELX, VX-445) in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects...” NCT04058353

“The purpose of this program is to provide elexacaftor(ELX, VX-445)/tezacaftor(TEZ)/ivacaftor(IVA) combination therapy to CF patients in critical need who are 12 years of age...” NCT04058210

“Following a run-in period of 4 weeks with Tezacaftor (TEZ)/Ivacaftor (IVA), participants received TEZ 100 milligram (mg)/IVA 150 mg as fixed-dose combination (FDC) tablet in...” NCT03460990

“This study will evaluate the pharmacokinetics (PK), safety, tolerability, efficacy, and pharmacodynamic effect of VX-659, tezacaftor (TEZ), and ivacaftor (IVA) when dosed in...” NCT03633526

“This is a Phase 2, randomized, double blind, placebo and active-controlled, parallel group, multicenter study designed to evaluate the safety and tolerability of VX-152 in...” NCT02951195

“This study will evaluate the long-term safety and tolerability of VX-659 in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects with cystic fibrosis...” NCT03447262

“This study will evaluate the efficacy of VX-659 in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects with cystic fibrosis (CF) who are heterozygous...” NCT03447249

“This study will evaluate the efficacy, safety, and pharmacodynamics of elexacaftor (ELX, VX-445) in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in...” NCT04105972

“Rationale: Elexacaftor/Tezacaftor/Ivacaftor (ELX/TEZ/IVA) was shown to be efficacious and safe in patients ≥12 years of age with cystic fibrosis and at least one F508del-CFTR...” PMID 33734030 Jun 2021

“The purpose of this study is to evaluate the long term safety, tolerability, efficacy and pharmacodynamics of elexacaftor (ELX)/tezacaftor (TEZ)/ivacaftor (IVA) in CF...” NCT05153317

“This study evaluated the long-term safety and tolerability of elexacaftor (ELX), tezacaftor (TEZ), and ivacaftor (IVA) triple combination (TC) treatment in participants with...” NCT04043806

“Participants received elexacaftor (ELX) 200 milligram (mg) once daily (qd)/tezacaftor (TEZ)100 mg qd/ivacaftor (IVA)150 mg every 12 hours (q12h) in the treatment period for 48 weeks.” NCT04362761

“Participants weighing less than (\<)40 kilograms (kg) at Day 1 received tezacaftor (TEZ) 50 milligrams (mg) once daily (qd)/ivacaftor (IVA) 75 mg every 12 hours (q12h)” NCT03537651

“The purpose of the study is to evaluate the long-term safety, tolerability, efficacy, and pharmacodynamics (PD) of elexacaftor (ELX)/tezacaftor (TEZ)/ivacaftor (IVA).” NCT06460506

“This study will evaluate the effects of elexacaftor/tezacaftor/ivacaftor (ELX/TEZ/IVA) on cough and physical activity using wearable technology in CF participants.” NCT04969224

“Participants who received lumacaftor (LUM, VX-809) 600 milligram (mg) plus ivacaftor (IVA, VX-770) 250 mg fixed-dose combination (FDC) tablet orally in the morning” NCT01931839

“This study will evaluate the efficacy of VX-445 in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects with cystic fibrosis (CF)” NCT03525548

“Lumacaftor (LUM) 200 mg every 12 hours (q12h)/ivacaftor (IVA) 250 mg q12h (for 6 through 11 years of age).” NCT02544451

“Trikafta (Elexacaftor \[ELX\], Tezacaftor \[TEZ\], Ivacaftor\[IVA\]) is contraindicated” NCT04840862

“it is combined with ivacaftor (IVA), an enhancer of the CFTR protein function.” NCT04581408

“VX-661 in combination with ivacaftor (IVA, VX-770) and IVA monotherapy” NCT02392234

“VX-661 (tezacaftor; TEZ) in combination with ivacaftor (IVA)” NCT02508207

“elexacaftor (ELX)/tezacaftor (TEZ)/ivacaftor (IVA)” NCT05111145

IVA (ivacaftor) 75 mg every 12 hours” NCT04183790

Ivacaftor (IVA) 150 mg tablet” NCT02070744

NCT03277196

Known as IVA, VX-770 IVA, VX-770NCT02392234
Known as Kalydeco “This is a prospective randomized double-blinded placebo-controlled crossover study of the short-term effects of ivacaftor (aka VX-770 or Kalydeco) on sweat chloride...” NCT01784419
4

“The new drug, Ivacaftor (KALYDECO), is a drug that has recently been approved by the U.S. Food and Drug Administration (FDA) for patients with a lung disease called Cystic...” NCT03251911

“All participants in group 7 who received placebo matched to VX-661 tablet orally qd in combination with physician-prescribed Kalydeco (Ivacaftor) for up to 28 days.” NCT01531673

NCT02599792

NCT02392702

Known as Orkambi ClinicalTrials.gov intervention name — accepted as the source's own label NCT02709109
Known as Symdeko ClinicalTrials.gov intervention name — accepted as the source's own label NCT03624101
Known as VX-770 “This is a prospective randomized double-blinded placebo-controlled crossover study of the short-term effects of ivacaftor (aka VX-770 or Kalydeco) on sweat chloride...” NCT01784419
16

“Combination treatment with the cystic fibrosis transmembrane conductance regulator (CFTR) modulators tezacaftor (VX-661) and ivacaftor (VX-770) was designed to target the...” PMID 29099344 Nov 2017

“The purpose of this study is to evaluate the effect of ivacaftor (VX-770) on lung clearance index (LCI) in subjects aged 6 years and older with cystic fibrosis (CF) who have...” NCT01262352

“Participants who received lumacaftor (LUM, VX-809) 600 milligram (mg) plus ivacaftor (IVA, VX-770) 250 mg fixed-dose combination (FDC) tablet orally in the morning” NCT01931839

“lumacaftor (VX-809), a CFTR corrector, in combination with ivacaftor (VX-770), a CFTR potentiator” PMID 25981758 May 2015

“Ivacaftor (VX-770), a cystic fibrosis transmembrane conductance regulator (CFTR) potentiator” PMID 23590265 Jun 2013

“VX-661 in combination with ivacaftor (IVA, VX-770) and IVA monotherapy” NCT02392234

“Ivacaftor (VX-770)” NCT03251911

NCT01208285

NCT01161537

NCT01381289

NCT01018368

NCT00966602

NCT01060566

NCT01153542

NCT02514473

NCT01216046

Action Activate “VX-770, a CFTR potentiator, has been shown to increase the activity of wild-type and defective cell-surface CFTR in vitro.” PMID 21083385 Nov 2010
Modality Small molecule “orally bioavailable small moleculeNCT01381289
Route Oral “receive oral VX-770 every 12 hours” PMID 21083385 Nov 2010
Target CFTR “Ivacaftor is a potent and selective CFTR potentiator of wild-type, G551D, F508del, and R117H forms of human CFTR protein.” NCT00457821