Drugs / Vintafolide
last change Nov 2016 re-read 2 minutes ago

Vintafolide

also known as EC145 · MK-8109 · Vintafolida

Other / unclassified targets FOLR1

Developed for
cancer · ovarian cancer · breast neoplasm · endometrial cancer · lung adenocarcinoma · non-small cell lung carcinoma
Investigated by
Endocyte

Trials 10 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 13 trials
Phase 1 NCT02049281 Feb → May 2014 cancer Endocyte Terminated No outcome recorded
Phase 1 NCT01688791 Dec 2012 → Sep 2014 Endocyte Terminated No outcome recorded
Phase 1 NCT00308269 Mar 2006 → Aug 2007 cancer Endocyte Completed No outcome recorded
Phase 26 trials
Phase 2 NCT01953536 Apr 2014 → Nov 2016 breast neoplasm Endocyte Withdrawn No outcome recorded
Phase 2 NCT01577654 Mar 2011 → Dec 2013 non-small cell lung carcinoma Endocyte Completed No outcome recorded
Phase 2 NCT01002924 Dec 2009 → Dec 2013 cancer Endocyte Completed No outcome recorded
Phase 2 NCT00722592 Sep 2008 → Sep 2010 ovarian cancer Endocyte Completed No outcome recorded
Phase 2 NCT00511485 Aug 2007 → Jul 2009 lung adenocarcinoma Endocyte Completed No outcome recorded
Phase 2 NCT00507741 Aug 2007 → Apr 2009 endometrial cancer, ovarian cancer Endocyte Completed No outcome recorded
Phase 31 trial
Phase 3 NCT01170650 Apr 2011 → May 2015 ovarian cancer Endocyte Terminated No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 12 sources stand behind the page.

FieldValueCited text
Known as vintafolide “Extension Study of EC145 (Vintafolide) for Subjects Enrolled in a Previous Study With EC145 (MK-8109-010)” NCT01002924
7

NCT00308269

NCT00511485

NCT00507741

NCT02049281

NCT00722592

NCT01688791

NCT01953536

Known as EC145 “Study of Vintafolide (MK-8109, EC145) in Participants With Advanced Ovarian and Endometrial Cancers (MK-8109-007, EC-FV-02)” NCT00507741
5

“Study of Vintafolide (MK-8109, EC145) in Participants With Progressive Adenocarcinoma of the Lung (MK-8109-008, EC-FV-03)” NCT00511485

“Study of Vintafolide (MK-8109, EC145) for the Treatment of Recurrent or Refractory Solid Tumors (MK-8109-006, EC-FV-01)” NCT00308269

NCT01577654

NCT01002924

NCT01170650

Known as MK-8109 “Study of Vintafolide (MK-8109, EC145) in Participants With Advanced Ovarian and Endometrial Cancers (MK-8109-007, EC-FV-02)” NCT00507741
2

“Study of Vintafolide (MK-8109, EC145) in Participants With Progressive Adenocarcinoma of the Lung (MK-8109-008, EC-FV-03)” NCT00511485

“Study of Vintafolide (MK-8109, EC145) for the Treatment of Recurrent or Refractory Solid Tumors (MK-8109-006, EC-FV-01)” NCT00308269

Known as Vintafolida ChEMBL registry synonym — accepted as the source's own label CHEMBL3039521
Modality Other / unclassified “EC145 (vintafolide), a conjugate of folic acid and the vinca alkaloid desacetylvinblastine hydrazide (DAVLBH)” PMID 23032618 Oct 2012
Route Intravenous “Vintafolide given by intravenous bolus or infusion” NCT00308269
Target FOLR1 “Folate receptor alpha binding agent” CHEMBL3039521