Drugs / Latrepirdine

Trials 28 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 112 trials
Phase 1 NCT00990613 Oct 2009 → Jan 2010 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00975481 Oct 2009 → Feb 2010 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00988624 Oct → Dec 2009 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00931073 Jul → Oct 2009 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00907322 Jun → Jul 2009 Pfizer Completed No outcome recorded
Phase 1 NCT00824590 Feb → Oct 2009 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00831506 Feb → May 2009 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00827034 Feb → Apr 2009 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00825084 Feb → May 2009 Alzheimer disease, Huntington disease Pfizer Completed No outcome recorded
Phase 1 NCT00831532 Feb → Aug 2009 liver failure Pfizer Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00387270 Oct 2006 → Mar 2007 Huntington disease Medivation, Inc. Completed No outcome recorded
Phase 25 trials
Phase 2 NCT06292351 Dec 2023 → Jan 2025 Alzheimer disease Bigespas LTD Completed No outcome recorded
Phase 2 NCT01066481 Apr 2010 → Mar 2012 Alzheimer disease Pfizer Withdrawn No outcome recorded
Phase 2 NCT00704782 Apr 2008 → Aug 2010 Alzheimer disease Medivation, Inc. Terminated No outcome recorded
Phase 2 NCT00497159 Jul 2007 → Jun 2008 Huntington disease Medivation, Inc. Completed No outcome recorded
Phase 2 NCT00377715 Sep 2005 → Aug 2006 Alzheimer disease Medivation, Inc. Completed No outcome recorded
Phase 310 trials
Phase 3 NCT01152216 Apr 2010 → May 2012 Alzheimer disease Medivation, Inc. Terminated No outcome recorded
Phase 3 NCT01066546 Apr → Jul 2010 Alzheimer disease Pfizer Terminated No outcome recorded
Phase 3 NCT01085266 Feb 2010 → Jun 2011 Huntington disease Medivation, Inc. Terminated No outcome recorded
Phase 3 NCT00954590 Oct 2009 → Aug 2010 Medivation, Inc. Terminated No outcome recorded
Phase 3 NCT00939783 Sep 2009 → Aug 2010 Alzheimer disease Pfizer Terminated No outcome recorded
Phase 3 NCT00912288 Sep 2009 → Aug 2010 Alzheimer disease Pfizer Terminated No outcome recorded
Phase 3 NCT00920946 Jul 2009 → Jul 2011 Huntington disease Medivation, Inc. Completed No outcome recorded
Phase 3 NCT00829374 Mar 2009 → Dec 2011 Alzheimer disease Medivation, Inc. Completed No outcome recorded
Phase 3 NCT00838110 Feb 2009 → Jan 2010 Alzheimer disease Pfizer Completed No outcome recorded
Phase 3 NCT00675623 May 2008 → Dec 2009 Alzheimer disease Medivation, Inc. Completed No outcome recorded

Evidence & citations 12 cited values

Every value below carries the sentence it was read from. 32 sources stand behind the page.

FieldValueCited text
Known as Latrepirdine Latrepirdine is an orally administered experimental small molecule that was initially developed as an antihistamine and subsequently was shown to stabilize mitochondrial...” PMID 23108692 Jan 2013
7

“A Phase 1, Fixed Sequence, Cross-Over Study To Investigate The Single Dose Pharmacokinetics Of A Dimebon (Latrepirdine) Transdermal Solution Relative To The Immediate Release...” NCT00990613

“An Open-Label Extension To The B1451006 Protocol To Evaluate The Safety And Efficacy Of Dimebon (Latrepirdine, PF-01913539) In Subjects With Moderate-To-Severe Alzheimer's Disease” NCT01066546

“A Study In Healthy Volunteers To Estimate The Pharmacokinetics Of Four Modified-Release Formulations Of Dimebon (Latrepirdine)” NCT00988624

“A Study To Evaluate The Abuse Potential Of Single Oral Doses Of Dimebon (Latrepirdine) In Healthy Recreational Polydrug Users” NCT00975481

“evaluate efficacy and safety of Latrepirdine polymorph DMB-I in 26-week” PMID 42141012 May 2026

“Dimebon (latrepirdine)” NCT01085266

“Dimebon (latrepirdine)” NCT00954590

Known as Dimebolin ChEMBL registry synonym — accepted as the source's own label CHEMBL589390
Known as Dimebolin dihydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL589390
Known as Dimebolin hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL589390
Known as Dimebon “B is oral doses of Dimebon 10 mg TID on Days 1 7 and Dimebon 20 mg TID on Days 8 17, with co administration of a single oral dose of warfarin 25 mg on Day 12 of the relevant...” NCT00827034
26

“DMB-I (Dimebon)” NCT06292351

NCT00497159

NCT00831532

NCT00387270

NCT00907322

NCT01152216

NCT00838110

NCT00824590

NCT00704782

NCT01066546

NCT00939783

NCT00829816

NCT00920946

NCT00377715

NCT00831506

NCT00954590

NCT00975481

NCT00825084

NCT00675623

NCT00931073

NCT00788047

NCT01085266

NCT00988624

NCT00912288

NCT00990613

NCT00829374

Known as Dimebon dihydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL589390
Known as DMB-I ClinicalTrials.gov intervention name — accepted as the source's own label NCT06292351
Known as Latrepirdina ChEMBL registry synonym — accepted as the source's own label CHEMBL589390
Known as LATREPIRDINE DIHYDROCHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL589390
Known as PF 01913539 “A Phase I, Open-Label, Three-Period, Fixed-Sequence Study To Estimate The Steady-State Effect Of Ketoconazole And Omeprazole On The Single-Dose Pharmacokinetics Of Dimebon...” NCT00931073
10

“A Phase 1, Randomized, Open-Label, Two-Way Crossover Study To Evaluate The Steady-State Effect Of Dimebon [PF-01913539] On The Single-Dose Pharmacokinetics Of The CYP2D6...” NCT00788047

“A Phase 3, Multi-Center, Randomized, Double-Blind Placebo-Controlled Study To Evaluate The Safety And Tolerability Of Dimebon (PF-01913539) For Up To 26-Weeks In Patients With...” NCT00838110

“A Phase 1, Randomized, Open-Label, Two-Way Crossover Study To Evaluate The Steady-State Effect Of Dimebon (PF 01913539) On The Single-Dose Pharmacokinetics And Pharmacodynamics...” NCT00827034

“A Phase 1, Non-Randomized, Open-Label, Single-Dose Study To Evaluate The Pharmacokinetics, Safety, And Tolerability Of Dimebon [PF 01913539] In Subjects With Severely-Impaired...” NCT00824590

“An Open-Label Extension To The B1451006 Protocol To Evaluate The Safety And Efficacy Of Dimebon (Latrepirdine, PF-01913539) In Subjects With Moderate-To-Severe Alzheimer's Disease” NCT01066546

“An Open Label Extension To The B1451027 Protocol To Evaluate The Long Term Safety And Tolerability Of Dimebon (PF 01913539) In Patients With Alzheimer's Disease” NCT00939783

“A Phase 1 Study To Evaluate The Pharmacokinetics, Safety, And Tolerability Of Dimebon [PF-01913539] In Japanese And Western Healthy Subjects” NCT00825084

“Dimebon (PF-01913539)-Digoxin Drug-Drug Interaction Study In Healthy Subjects” NCT00831506

“Dimebon [Pf-01913539]” NCT00831532

NCT01066481

Modality Small molecule “Latrepirdine is an orally administered experimental small moleculePMID 23108692 Jan 2013
Route Oral “receive oral dimebon, 20 mg three times a day” PMID 18640457 Jul 2008