Drugs / Tavapadon
last change Dec 2025 re-read 2 minutes ago

Tavapadon

also known as PF-06649751 · CVL-751

Small molecule targets DRD1, DRD5 via activation

Developed for
Parkinson disease
Investigated by
Pfizer · AbbVie · Cerevel Therapeutics, LLC

Trials 19 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 112 trials
Phase 1 NCT06895356 Mar → Jun 2025 AbbVie Completed No outcome recorded
Phase 1 NCT05581823 Oct 2022 → Jan 2023 Parkinson disease Cerevel Therapeutics, LLC Completed No outcome recorded
Phase 1 NCT05404542 May 2022 → Aug 2023 impaired renal function disease Cerevel Therapeutics, LLC Completed No outcome recorded
Phase 1 NCT05404529 Apr 2022 → Jan 2023 liver disease, severe congenital Cerevel Therapeutics, LLC Completed No outcome recorded
Phase 1 NCT04241393 Feb → Nov 2020 Cerevel Therapeutics, LLC Completed No outcome recorded
Phase 1 NCT04295642 Jan 2020 → Jul 2021 Parkinson disease Cerevel Therapeutics, LLC Completed No outcome recorded
Phase 1 NCT03121664 Apr → Sep 2017 Pfizer Completed No outcome recorded
Phase 1 NCT02373072 Mar 2015 → Feb 2016 Parkinson disease Pfizer Completed No outcome recorded
Phase 1 NCT02262767 Nov → Dec 2014 Pfizer Completed No outcome recorded
Phase 1 NCT02224664 Oct 2014 → Mar 2016 Parkinson disease Pfizer Completed No outcome recorded
Phase 23 trials
Phase 2 NCT03185481 Jul → Oct 2017 Parkinson disease Pfizer Terminated No outcome recorded
Phase 2 NCT02847650 Oct 2016 → Jan 2018 Parkinson disease Pfizer Terminated No outcome recorded
Phase 2 NCT02687542 Mar 2016 → Nov 2017 Parkinson disease Pfizer Terminated No outcome recorded
Phase 34 trials
Phase 3 NCT04760769 Feb 2021 → Dec 2025 Parkinson disease AbbVie Completed No outcome recorded
Phase 3 NCT04542499 Sep 2020 → Jan 2024 Parkinson disease AbbVie Completed No outcome recorded
Phase 3 NCT04223193 Jan 2020 → Oct 2024 Parkinson disease AbbVie Completed No outcome recorded
Phase 3 NCT04201093 Dec 2019 → Jun 2024 Parkinson disease AbbVie Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
NCT07158827 Background Parkinson disease AbbVie Available No outcome recorded

Press releases naming this drug 10 releases

DateIssuerRelease
2025-09-26 AbbVie AbbVie Submits New Drug Application to U.S. FDA for Tavapadon for the Treatment of Parkinson's Disease abbvie.com
2024-12-09 AbbVie AbbVie Announces Positive Topline Results for the Phase 3 TEMPO-2 Trial Evaluating Tavapadon as a Monotherapy for Parkinson's Disease abbvie.com
2024-09-26 AbbVie AbbVie Announces Positive Topline Results from Phase 3 TEMPO-1 Trial Evaluating Tavapadon as a Monotherapy for Parkinson's Disease abbvie.com
2024-04-18 AbbVie Cerevel Therapeutics Announces Positive Topline Results for Tavapadon in Phase 3 Adjunctive Trial for People Living with Parkinson’s Disease abbvie.com
2023-11-29 AbbVie Cerevel Therapeutics to Host Investor Webcast on Tavapadon in Parkinson’s Disease abbvie.com
2021-04-13 AbbVie Cerevel Therapeutics Announces Strategic $125 Million Non-Dilutive Financing Transaction for Tavapadon abbvie.com
2020-10-30 AbbVie Cerevel Therapeutics Announces First Patients Dosed in all Phase 3 Trials of Tavapadon for the Treatment of Parkinson’s Disease abbvie.com
2020-01-14 AbbVie Cerevel Therapeutics Initiates Phase 3 Program of Tavapadon for the Treatment of Parkinson’s Disease abbvie.com
2019-09-23 AbbVie Cerevel Therapeutics Announces Positive Results from a Phase 2 Study of Tavapadon in Patients with Early-stage Parkinson’s Disease abbvie.com
2019-09-19 AbbVie Cerevel Therapeutics to Present Results from a Phase 2 Study of Tavapadon in Patients with Early-stage Parkinson’s Disease abbvie.com

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 22 sources stand behind the page.

FieldValueCited text
Known as Tavapadon ClinicalTrials.gov intervention name — accepted as the source's own label NCT06895356
9

NCT05404529

NCT04241393

NCT04542499

NCT05404542

NCT04223193

NCT04201093

NCT04760769

NCT05581823

NCT07158827

Known as CVL-751 ClinicalTrials.gov intervention name — accepted as the source's own label NCT04295642
Known as PF-06649751 ClinicalTrials.gov intervention name — accepted as the source's own label NCT02687542
8

NCT03185481

NCT02262767

NCT03121664

NCT01981694

NCT02847650

NCT02224664

NCT02373072

NCT02066909

Action Activate “PF-06649751 is a novel, highly selective dopamine D1/D5 agonist targeted for Parkinson's disease treatment.” PMID 30361858 Oct 2018
2

“Dopamine D5 receptor partial agonist” CHEMBL3697617

“Dopamine D1 receptor partial agonist” CHEMBL3697617

Modality Small molecule CHEMBL3697617
Route Oral “given orally” NCT01981694
Target DRD1 “Dopamine D1 receptor partial agonist” CHEMBL3697617
Target DRD5 “Dopamine D5 receptor partial agonist” CHEMBL3697617