drugset / Trial / NCT02253420

COPANLISIB (BAY80-6946) Drug-drug Interaction and Cardiovascular Safety Study in Advanced Solid Tumor and Non-Hodgkin's Lymphoma Patients

NCT02253420

Phase 1 Completed 51 enrolled Bayer
Non-randomizedSingle-groupOpen-labelOther

Summary

To evaluate the effect of itraconazole or rifampin on the absorption, distribution, metabolism and elimination of COPANLISIB (BAY80-6946). To evaluate the effect of copanlisib on QT/QTc intervals and left ventricular ejection fraction as parameters of cardiovascular safety.

Timeline

Start
2014-10-08
Primary completion
2018-03-12
Completion
2019-08-13

Drugs

EvaluationDrugModalityDoseRoute
Subject Copanlisib Small molecule 12 mg Intravenous
Subject Copanlisib Small molecule 30 mg Intravenous
Subject Copanlisib Small molecule 60 mg Intravenous
Subject Itraconazole Small molecule 200 mg Oral
Subject Rifampin Small molecule 600 mg Oral

Indications

No indication recorded.