drugset / Trial / NCT03561298

A Pharmacokinetic Study to Assess Drug-drug Interaction Between Zanubrutinib and a Cocktail of Substrates in Healthy Subjects

NCT03561298

Phase 1 Completed 18 enrolled BeiGene
NaSingle-groupOpen-labelTreatment

Summary

This study is designed to evaluate the safety and pharmacokinetic interaction of effects of multiple doses of zanubrutinib with a "Cocktail" of five probe drugs for cytochrome P450 (CYP) 3A, CYP2C9, CYP2C19, P-glycoprotein and breast cancer resistance protein (BCRP) in healthy subjects

Timeline

Start
2018-06-07
Primary completion
2018-06-07
Completion
2018-07-02

Drugs

EvaluationDrugModalityDoseRoute
Subject Digoxin Other / unclassified
Subject Midazolam Small molecule
Subject Omeprazole Other / unclassified
Subject Rosuvastatin Small molecule
Subject Warfarin Small molecule
Subject Zanubrutinib Small molecule

Indications

No indication recorded.