drugset / Trial / NCT05176483

Study of Zanzalintinib in Combination With Immuno-Oncology Agents in Participants With Solid Tumors

NCT05176483

Phase 1 Recruiting 1314 enrolled Exelixis
Non-randomizedSequentialOpen-labelTreatment

Summary

This is a multicenter Phase 1b, open label, dose-escalation and cohort-expansion study, evaluating the safety, tolerability, pharmacokinetics (PK), preliminary antitumor activity, and effect of biomarkers of zanzalintinib administered alone, and in combination with nivolumab (doublet), nivolumab + ipilimumab (triplet) and nivolumab + relatlimab (triplet) in participants with advanced solid tumors. In the Expansion Stage, the safety and efficacy of zanzalintinib as monotherapy and in combination therapy will be further evaluated in tumor-specific Expansion Cohorts.

Timeline

Start
2021-12-14
Primary completion
2030-06-28
Completion
2030-06-28

Drugs

EvaluationDrugModalityDoseRoute
Subject Ipilimumab Monoclonal antibody 1 mg/kg Intravenous
Subject Nivolumab Monoclonal antibody 360 mg Intravenous
Subject Nivolumab Monoclonal antibody 480 mg Intravenous
Subject Nivolumab Monoclonal antibody Intravenous
Subject Relatlimab Monoclonal antibody Intravenous
Subject Zanzalintinib Small molecule Oral