drugset / Trial / NCT07349537

Study of RMC-5127 in Patients With Advanced KRAS G12V-Mutant Solid Tumors

NCT07349537

Phase 1 Recruiting 574 enrolled Revolution Medicines, Inc.
Non-randomizedParallel-groupOpen-labelTreatment

Summary

The purpose of this study is to evaluate the safety, tolerability, pharmacokinetics (PK), and preliminary antitumor activity of RMC-5127 as a monotherapy and in combination with either daraxonrasib or cetuximab in adults with KRAS G12V-mutant solid tumors.

Timeline

Start
2026-01-08
Primary completion
2028-04
Completion
2028-10

Drugs

EvaluationDrugModalityDoseRoute
Subject Cetuximab Monoclonal antibody Intravenous
Subject RMC-5127 Unknown Oral
Subject daraxonrasib Small molecule Oral