Drugs / Lersivirine
last change Apr 2013 re-read 2 minutes ago

Lersivirine

also known as UK 453,061 · Lersivirina

Small molecule

Investigated by
Pfizer · ViiV Healthcare

Trials 9 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 15 trials
Phase 1 NCT01603485 Jun → Aug 2012 Pfizer Completed No outcome recorded
Phase 1 NCT01220232 Nov 2010 → Jan 2011 Pfizer Completed No outcome recorded
Phase 1 NCT01099748 May → Jun 2010 Pfizer Completed No outcome recorded
Phase 1 NCT00925535 May → Aug 2010 Pfizer Completed No outcome recorded
Phase 1 NCT00936871 Jan → Mar 2010 Pfizer Completed No outcome recorded
Phase 24 trials
Phase 2 NCT01254656 Feb 2011 → Apr 2013 Pfizer Terminated No outcome recorded
Phase 2 NCT00823979 Mar 2009 → Oct 2012 Pfizer Terminated No outcome recorded
Phase 2 NCT00824421 Feb 2009 → Oct 2011 Pfizer Completed No outcome recorded
Phase 2 NCT00348673 Feb 2006 → Feb 2007 Pfizer Completed No outcome recorded
Also used as a comparator or background therapy in 3 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1 NCT01230385 Comparator Oct 2010 → May 2011 Pfizer Completed No outcome recorded
Phase 1 NCT01050751 Comparator Feb → Mar 2010 Pfizer Completed No outcome recorded
Phase 1 NCT00784420 Comparator Sep → Nov 2008 Pfizer Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 13 sources stand behind the page.

FieldValueCited text
Known as Lersivirine ClinicalTrials.gov intervention name — accepted as the source's own label NCT01099748
7

NCT01050751

NCT00936871

NCT01254656

NCT01220232

NCT01603485

NCT00925535

NCT01230385

Known as Lersivirina ChEMBL registry synonym — accepted as the source's own label CHEMBL571987
Known as UK 453,061 “Open-Label, Randomized, 2-Way Crossover Study To Estimate The Pharmacokinetics And Bioavailability Of Lersivirine (UK 453,061) Administered As A Single 750 Mg Tablet And 3 X...” NCT01050751
8

“A Phase 1, Randomized, Single Dose, Placebo And Active Controlled, 3-Way Crossover Study To Evaluate The Effect Of A Single Oral Dose Of Lersivirine (UK-453,061) On Qt...” NCT00936871

“Open-Label, Randomized, Crossover Study to Estimate the Pharmacokinetics, Bioavailability and Effect of Food on Single Dose Modified-release Lersivirine (UK-453,061) 500 mg in...” NCT01603485

“Open Label, Single-Sequence Study To Estimate The Effect Of Lersivirine (UK-453,061) On S- And R-Methadone In Subjects Receiving Chronic Methadone Treatment” NCT01099748

“UK-453,061 500 mg tablets PO QD + Tenofovir DF 300 mg/Emtricitabine 200 mg tablets PO QD.” NCT00824421

“Drug Interaction Study Between Rifabutin And Lersivirine (UK-453,061)” NCT00925535

NCT00784420

NCT00823979

NCT00348673

Modality Small molecule CHEMBL571987
Route Oral “UK-453,061 500 mg tablets PO QD” NCT00824421