Drugs / AZD1386
last change Jan 2013 re-read 9 days ago

AZD1386

Small molecule targets TRPV1 via inhibition

Developed for
chronic pain syndrome · esophageal disorder · neuropathy, painful
Investigated by
AstraZeneca

Trials 11

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 17 trials
Phase 1 NCT00945178 Aug → Sep 2009 — AstraZeneca Terminated No outcome recorded
Phase 1 NCT00832169 Jan → Feb 2009 — AstraZeneca Completed No outcome recorded
Phase 1 NCT00711048 Jun 2008 → Jul 2009 — AstraZeneca Completed No outcome recorded
Phase 1 NCT00714337 Jun → Aug 2008 — AstraZeneca Completed No outcome recorded
Phase 1 NCT00736658 Jun → Sep 2008 chronic pain syndrome AstraZeneca Completed No outcome recorded
Phase 1 NCT00690079 Feb → Oct 2008 chronic pain syndrome AstraZeneca Completed No outcome recorded
Phase 1 NCT00692146 Jan → May 2008 — AstraZeneca Completed No outcome recorded
Phase 24 trials · 2 missed
Phase 2 NCT01019928 Nov 2009 → Jan 2011 esophageal disorder AstraZeneca Completed Missed primary
Phase 2 NCT00976534 Sep 2009 → Feb 2010 neuropathy, painful AstraZeneca Terminated No outcome recorded
Phase 2 NCT00878501 Mar → Jul 2009 — AstraZeneca Terminated Missed primary
Phase 2 NCT00672646 Apr → Jun 2008 — AstraZeneca Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 14 sources stand behind the page.

FieldValueCited text
Known as AZD1386 ClinicalTrials.gov intervention name — accepted as the source's own label NCT00711048 ↗
10

NCT01019928 ↗

NCT00832169 ↗

NCT00976534 ↗

NCT00714337 ↗

NCT00945178 ↗

NCT00692146 ↗

NCT00878501 ↗

NCT00672646 ↗

NCT00690079 ↗

NCT00736658 ↗

Action Inhibit “AIM: To investigate the effect of a TRPV1 antagonist (AZD1386) on experimentally induced oesophageal pain.” PMID 21410733 ↗ Mar 2011
Modality Small molecule — CHEMBL3545039 ↗
Route Oral “95mg, oral solution, single dose” NCT00672646 ↗
Target TRPV1 “TRPV1 antagonist AZD1386” PMID 23320520 ↗ Jan 2013