Drugs / GFH375
last change Jul 2026 re-read 2 minutes ago

GFH375

Small molecule targets KRAS via inhibition

Developed for
malignant pancreatic neoplasm · non-small cell lung carcinoma · cancer · colorectal cancer · pancreatic ductal adenocarcinoma
Investigated by
Genfleet Therapeutics (Shanghai) Inc.

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/22 trials
Phase 1/2 NCT07259590 Oct 2025 → Jul 2027 expected colorectal cancer, pancreatic ductal adenocarcinoma Genfleet Therapeutics (Shanghai) Inc. Recruiting No outcome recorded
Phase 1/2 NCT06500676 Jul 2024 → Jul 2028 expected cancer Genfleet Therapeutics (Shanghai) Inc. Recruiting No outcome recorded
Phase 22 trials
Phase 2 NCT07554859 May 2026 → Apr 2027 expected non-small cell lung carcinoma Genfleet Therapeutics (Shanghai) Inc. Not yet recruiting No outcome recorded
Phase 2 NCT07026916 Aug 2025 → Aug 2027 malignant pancreatic neoplasm Genfleet Therapeutics (Shanghai) Inc. Withdrawn No outcome recorded
Phase 32 trials
Phase 3 NCT07668752 Jul 2026 → Jun 2030 expected non-small cell lung carcinoma Genfleet Therapeutics (Shanghai) Inc. Not yet recruiting No outcome recorded
Phase 3 NCT07262567 Dec 2025 → Jun 2027 expected malignant pancreatic neoplasm Genfleet Therapeutics (Shanghai) Inc. Recruiting No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 6 sources stand behind the page.

FieldValueCited text
Known as GFH375 ClinicalTrials.gov intervention name — accepted as the source's own label NCT06500676
5

NCT07026916

NCT07668752

NCT07554859

NCT07262567

NCT07259590

Action Inhibit “GFH375 is an oral, highly selective, non-covalent small-molecule inhibitor targeting the KRAS G12D mutation.” NCT07668752
Modality Small molecule “GFH375 is an oral, highly selective, non-covalent small-molecule inhibitor targeting the KRAS G12D mutation.” NCT07668752
Route Oral orally” NCT06500676
Target KRAS “targeting the KRAS G12D mutation” NCT07668752